SCHEMBL28053244

SCHEMBL28053244

NS(=O)(=O)c1ccc(OC(F)(F)F)c(-c2cncc(Cl)c2O)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.44
ALPL P05186 3/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
CA2 P00918 3/20 0.36
PTGS1 P23219 4/20 0.36
PTGS2 P35354 4/20 0.36
CA1 P00915 2/20 0.35
CA9 Q16790 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053258 0.81 PKM (0.46) CA2PTGS1PTGS2CA1CA9
SCHEMBL28053374 0.78 LRRK2 (0.44) CA2PTGS1PTGS2CA1CA9
SCHEMBL16235371 0.71 S100A9 (0.58) ALPLCYP2C9CYP2C19
SCHEMBL28053242 0.70 APLNR (0.43) CA2PTGS1PTGS2CA1CA9
SCHEMBL28053327 0.70 APLNR (0.45) CA2PTGS1PTGS2CA1CA9
SCHEMBL28826183 0.70 APLNR (0.40) CA2PTGS1PTGS2CA1CA9
SCHEMBL1081818 0.69 RORC (0.49) RORCSLC6A4SLC6A3CA2PTGS1
SCHEMBL28053322 0.69 APLNR (0.51) CA2PTGS1PTGS2CA1CA9
SCHEMBL28053239 0.68 APLNR (0.38) RORCCA2PTGS1PTGS2CA1
SCHEMBL28826194 0.68 SOS1 (0.39) CA2CA1CA9CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN claimed
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed