SCHEMBL28053347

SCHEMBL28053347

NS(=O)(=O)c1ccc(-c2cncc(Cl)c2O)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 10/20 0.44
CA2 P00918 10/20 0.44
CA9 Q16790 9/20 0.44
CA12 O43570 7/20 0.44
CA4 P22748 3/20 0.44
CA5A P35218 3/20 0.44
CA7 P43166 3/20 0.44
CA14 Q9ULX7 3/20 0.44
CA6 P23280 2/20 0.44
CA13 Q8N1Q1 2/20 0.44
VRK2 Q86Y07 1/20 0.38
PTGS2 P35354 2/20 0.33
ALOX5AP P20292 2/20 0.33
FEN1 P39748 2/20 0.33
PTGS1 P23219 1/20 0.33
APLNR P35414 1/20 0.33
RPS6KA3 P51812 1/20 0.31
CA5B Q9Y2D0 1/20 0.31
IKBKB O14920 1/20 0.31
CHUK O15111 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053327 0.76 APLNR (0.45) CA1CA2CA9CA12CA4
SCHEMBL28053322 0.75 APLNR (0.51) CA1CA2CA9CA12CA4
SCHEMBL28053258 0.71 PKM (0.46) CA1CA2CA9CA12CA4
SCHEMBL2704697 0.68 CA1 (0.61) CA1CA2CA9CA12CA4
SCHEMBL28053234 0.68 NPSR1 (0.41) CA1CA2CA9CA12
SCHEMBL28053374 0.68 LRRK2 (0.44) CA1CA2CA9CA12CA4
SCHEMBL28053242 0.68 APLNR (0.43) CA1CA2CA9VRK2PTGS2
SCHEMBL28826183 0.65 APLNR (0.40) CA1CA2CA9CA12CA4
SCHEMBL8974338 0.65 CA1 (0.44) CA1CA2CA9CA12CA4
SCHEMBL8652736 0.65 PTGS2 (0.63) CA1CA2CA9CA12CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed