SCHEMBL28077397

SCHEMBL28077397

Cc1ccc(-c2nc(O)c(O)s2)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.37
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
ALOX5 P09917 2/20 0.36
MAP3K5 Q99683 1/20 0.35
APP P05067 1/20 0.35
S1PR1 P21453 2/20 0.34
S1PR3 Q99500 1/20 0.34
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
HPGD P15428 1/20 0.33
CASP3 P42574 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28077207 0.78 ALDH1A1 (0.46) ALOX5S1PR1MAPTKDM4ESMN1; SMN2
SCHEMBL28077336 0.77 HDAC9 (0.39) ESR1ESR2ALOX5MAPT
SCHEMBL6842692 0.74 TP53 (0.39) GRM2MAP3K5S1PR1S1PR3MAPT
SCHEMBL13072194 0.73 RAB9A (0.50) MAPTKDM4EPOLBHPGDCASP3
SCHEMBL28831015 0.72 ALOX5 (0.62) ALOX5KDM4E
SCHEMBL6838624 0.71 TP53 (0.38) MAP3K5S1PR1S1PR3MAPTKDM4E
SCHEMBL28077372 0.70 SLC9A1 (0.35) ALOX5MAPTKDM4EHPGDSMN1; SMN2
SCHEMBL28077481 0.70 TRPM8 (0.53) ALOX5
SCHEMBL16806044 0.70 ALOX5 (0.47) GRM2ALOX5APPMAPTKDM4E
SCHEMBL13520606 0.70 GRM2 (0.44) GRM2ESR1ESR2HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104334544-B Benzimidazole proline derivative 埃科特莱茵药品有限公司 2016-10-19 CN disclosed