SCHEMBL28209158

SCHEMBL28209158

FC(F)(F)c1ccc(-c2cccnn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.50
TOP1 P11387 3/20 0.46
NPC1 O15118 1/20 0.45
MAOB P27338 1/20 0.43
TRPV1 Q8NER1 1/20 0.42
NPY5R Q15761 1/20 0.42
HDAC4 P56524 2/20 0.40
DHODH Q02127 1/20 0.40
NISCH Q9Y2I1 1/20 0.40
SCN2A Q99250 2/20 0.39
TGFBR1 P36897 1/20 0.39
S1PR1 P21453 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23258136 0.81 KIF11 (0.50) KIF11NPC1TRPV1HDAC4DHODH
SCHEMBL28289136 0.80 CTSS (0.53) MAOBNPY5RSCN2A
SCHEMBL3458918 0.78 NPY5R (0.47) TOP1NPC1MAOBNPY5RHDAC4
SCHEMBL28210972 0.78 NPY5R (0.42) KIF11NPC1NPY5R
SCHEMBL1456246 0.77 MAPT (0.46) NPC1HDAC4DHODH
SCHEMBL28211564 0.77 SCN5A (0.49) NPC1NPY5RNISCHSCN2A
SCHEMBL26135623 0.77 NPSR1 (0.43) KIF11NPC1TRPV1NPY5R
SCHEMBL13458062 0.75 GABRA1 (0.52) NPC1HDAC4DHODH
SCHEMBL28211548 0.75 TRPV4 (0.43)
SCHEMBL121970 0.74 RAB9A (0.50) NPC1HDAC4DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106458952-B Heterocycle sulfamide derivatives and drug containing the heterocycle sulfamide derivatives EA制药株式会社 2019-09-27 CN disclosed
CN-106061974-B Maleimide derivatives as the conditioning agent of WNT approach 新加坡科技研究局 2018-04-20 CN disclosed
CN-107849029-A Cyclopropane derivatives and drugs containing the same EA制药株式会社 2018-03-27 CN disclosed