SCHEMBL28292621

SCHEMBL28292621

NC(=O)Oc1ccnc(C(=O)NCCO)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.46
RAF1 P04049 1/20 0.44
S1PR1 P21453 1/20 0.42
KMT2A Q03164 3/20 0.41
MEN1 O00255 1/20 0.41
P2RX3 P56373 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
SPHK2 Q9NRA0 1/20 0.38
SPHK1 Q9NYA1 1/20 0.38
MMP13 P45452 1/20 0.38
ACR P10323 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28292627 0.87 SCN9A (0.41) BRAFRAF1KMT2AMEN1LOXL2
SCHEMBL28294334 0.82 LOXL2 (0.46) RAF1KMT2AMEN1LOXL2
SCHEMBL28940983 0.81 SCN9A (0.40) BRAFRAF1KMT2AMEN1LOXL2
SCHEMBL28963812 0.81 SCN9A (0.40) BRAFRAF1KMT2AMEN1LOXL2
SCHEMBL28292592 0.81 KDR (0.53) BRAFRAF1KMT2AMEN1
SCHEMBL20292453 0.80 BRAF (0.53) BRAFRAF1P2RX3MMP13
SCHEMBL28292566 0.78 MAOB (0.49) MAPTMMP13
SCHEMBL28292634 0.78 MEN1 (0.52) BRAFRAF1KMT2AMEN1ALDH1A1
SCHEMBL8945361 0.78 ITGB3 (0.44) S1PR1KMT2AMEN1LOXL2SMN1; SMN2
SCHEMBL6014835 0.77 MMP13 (0.64) BRAFRAF1KMT2AMEN1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN claimed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed