SCHEMBL28293162

SCHEMBL28293162

CS(=O)(=O)Nc1cccc2[nH]c(CCOC=O)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.46
JAK1 P23458 1/20 0.46
PARP14 Q460N5 5/20 0.43
MTNR1A P48039 3/20 0.40
MTNR1B P49286 3/20 0.40
KEAP1 Q14145 2/20 0.40
MCL1 Q07820 3/20 0.35
NFE2L2 Q16236 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ALOX15 P16050 1/20 0.34
HTT P42858 1/20 0.34
GLO1 Q04760 1/20 0.34
NR3C1 P04150 1/20 0.34
PGR P06401 1/20 0.34
NR3C2 P08235 1/20 0.34
AR P10275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27491895 0.78 DAO (0.43) MTNR1AMTNR1BMCL1NR3C1PGR
SCHEMBL27906754 0.77 DAO (0.44) MTNR1AMTNR1BKDM4EALDH1A1HPGD
SCHEMBL28168776 0.77 FBP1 (0.48) MTNR1AMTNR1BKDM4EHSD17B10HTT
SCHEMBL28678160 0.76 MTNR1A (0.58) MTNR1AMTNR1BKDM4ESMN1; SMN2HTT
SCHEMBL28880746 0.76 PTGS2 (0.45) MTNR1AMTNR1BALDH1A1
SCHEMBL27965811 0.76 PARP1 (0.40) MTNR1AMTNR1B
SCHEMBL27524233 0.76 DAO (0.43) MTNR1AMTNR1BKDM4EHPGD
SCHEMBL28291608 0.75 MMP2 (0.50) MTNR1AMTNR1BKDM4EALDH1A1HPGD
SCHEMBL28293142 0.75 MMP2 (0.40) MTNR1AMTNR1BKDM4EALDH1A1HPGD
SCHEMBL28291601 0.74 MTNR1A (0.38) MTNR1AMTNR1BKDM4EALDH1A1NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109748840-A A kind of synthetic method of 2- substituted indole derivative 中国医学科学院药物研究所 2019-05-14 CN disclosed