SCHEMBL283280

SCHEMBL283280

CCOC(=O)c1nnc(N)s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.52
HPGD P15428 4/20 0.52
MAPT P10636 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
GAA P10253 2/20 0.52
CYP1A2 P05177 2/20 0.51
POLB P06746 1/20 0.50
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
HTT P42858 2/20 0.49
TSHR P16473 1/20 0.49
FHIT P49789 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 2/20 0.44
HSD17B10 Q99714 3/20 0.43
MAPK1 P28482 2/20 0.42
ALOX15 P16050 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAOA P21397 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13800984 0.86 MAPT (0.44) ALDH1A1HPGDMAPTSMN1; SMN2GAA
SCHEMBL13800905 0.83 LMNA (0.47) ALDH1A1MAPTSMN1; SMN2GAACYP1A2
SCHEMBL299130 0.81 ALDH1A1 (0.46) ALDH1A1HPGDMAPTSMN1; SMN2GAA
SCHEMBL4315953 0.81 ALDH1A1 (0.46) ALDH1A1HPGDMAPTSMN1; SMN2GAA
SCHEMBL13800973 0.81 ALDH1A1 (0.42) ALDH1A1MAPTSMN1; SMN2GAACYP1A2
SCHEMBL12536605 0.81 ALDH1A1 (0.44) ALDH1A1HPGDMAPTSMN1; SMN2GAA
SCHEMBL368639 0.79 HSD17B10 (0.50) ALDH1A1HPGDMAPTSMN1; SMN2POLB
SCHEMBL24369643 0.78 ALDH1A1 (0.43) ALDH1A1HPGDMAPTSMN1; SMN2GAA
SCHEMBL281865 0.78 MAPT (0.43) ALDH1A1HPGDMAPTSMN1; SMN2GAA
SCHEMBL15945408 0.78 GAA (0.50) ALDH1A1HPGDMAPTSMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 255 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024245310-A1 THIAZOLYL OR THIADIAZOLYL AMIDES DERIVATIVES AND USE THEREOF NINGBO NEWBAY TECHNOLOGY DEVELOPMENT CO., LTD. (CN) 2024-12-05 WO disclosed
CN-118994142-A Furanamide compound and application thereof 浙江大学金华研究院 2024-11-22 CN disclosed
US-11993591-B2 Chromen-4-one derivatives for the treatment and prophylaxis of hepatitis B virus disease HOFFMANN-LA ROCHE INC. (US) 2024-05-28 US disclosed
CN-118084937-A Bicyclic heteroaromatic ring derivatives 杏林制药株式会社 2024-05-28 CN disclosed
US-11952387-B2 Bicyclic heteroaromatic ring derivative KYORIN PHARMACEUTICAL CO., LTD (JP) 2024-04-09 US disclosed
CN-112752761-B Bicyclic heteroaromatic ring derivatives 杏林制药株式会社 2024-03-29 CN disclosed
US-20230270750-A1 CARBALDEHYDE OXIMES AS BUTYRYLCHOLINESTERASE REACTIVATORS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2023-08-31 US disclosed
WO-2023152182-A1 NOVEL COMPOUNDS MODULATING MIR-155 SAVERNA THERAPEUTICS AG (CH) 2023-08-17 WO disclosed
US-11713313-B2 GLS1 inhibitors for treating disease BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-08-01 US disclosed
US-11713313-B2 GLS1 inhibitors for treating disease BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2023-08-01 US disclosed
WO-2008021926-A2 MODULATORS OF GLUCOCORTICOID RECEPTOR, AND/OR AP-1, AND/OR NF-KB ACTIVITY AND USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2008-02-21 WO disclosed
WO-2007038865-A1 SUBSTITUTED QUINOLINES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA LTD. (CA) 2007-04-12 WO disclosed
US-20070054897-A1 1,1-Dicyclohexyl-3-thiazol-2-yl-urea, 3-(5-Chloro-thiazol-2-yl)-1,1-dicyclohexyl-urea, for example; useful for the management, treatment, control, or adjunct treatment of diseases, where increasing glucokinase activity is beneficial, in particular, type 2 diabetes NOVO NORDISK A/S (DK) 2007-03-08 US disclosed
CN-1910166-A Heteroaryl ureas and their use as glucokinase activators NOVO NORDISK AS (DK) 2007-02-07 CN disclosed
WO-2007006814-A1 UREA GLUCOKINASE ACTIVATORS NOVO NORDISK A/S (DK) 2007-01-18 WO disclosed
EP-1723128-A1 HETEROARYL-UREAS AND THEIR USE AS GLUCOKINASE ACTIVATORS NOVO NORDISK A/S (DK) 2006-11-22 EP disclosed
WO-2005066145-A1 HETEROARYL-UREAS AND THEIR USE AS GLUCOKINASE ACTIVATORS NOVO NORDISK A/S (DK) 2005-07-21 WO disclosed
EP-0581502-B1 Antibiotic carbapenem compounds ZENECA LTD (GB) 1998-10-21 EP disclosed
US-5527793-A Antibiotic carbapenem compounds ZENECA LIMITED (GB) 1996-06-18 US disclosed
EP-0581502-A1 Antibiotic carbapenem compounds ZENECA LIMITED (GB) 1994-02-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11952387-B2 Bicyclic heteroaromatic ring derivative ZC3HAV1, RNASEH1, HAVCR2 ALDH1A1 1471/4885HPGD 3340/4885MAPT 2437/4885
US-11993591-B2 Chromen-4-one derivatives for the treatment and prophylaxis of hepatitis B virus disease HAVCR2, CYP7A1, CYP26B1 ALDH1A1 629/4885HPGD 1713/4885MAPT 3644/4885
US-20230270750-A1 CARBALDEHYDE OXIMES AS BUTYRYLCHOLINESTERASE REACTIVATORS BCHE, ACHE, CHAT ALDH1A1 239/4885HPGD 374/4885MAPT 2056/4885
US-11713313-B2 GLS1 inhibitors for treating disease GLS2, GLS, GLG1 ALDH1A1 882/4885HPGD 570/4885MAPT 4200/4885
US-20070054897-A1 1,1-Dicyclohexyl-3-thiazol-2-yl-urea, 3-(5-Chloro-thiazol-2-yl)-1,1-dicyclohexyl-urea, for example; useful for the management, treatment, control, or adjunct treatment of diseases, where increasing glucokinase activity is beneficial, in particular, type 2 diabetes GCK, GCKR, HK1 ALDH1A1 520/4885HPGD 1486/4885MAPT 2414/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.