SCHEMBL28344530

SCHEMBL28344530

N#Cc1cccc(C(=O)[O-])c1C#N.[Na+]

nearest known ligand 0.44

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 known ✓ P00915 3/20 0.40
CA2 known ✓ P00918 3/20 0.40
IKBKB O14920 3/20 0.44
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 1/20 0.42
POLB P06746 2/20 0.36
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
NOTUM Q6P988 1/20 0.34
SLC22A12 Q96S37 2/20 0.34
SLC22A6 Q4U2R8 1/20 0.34
SLC2A9 Q9NRM0 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34
GAA P10253 1/20 0.33
CXCR2 P25025 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11120196 0.82 POLB (0.38) KDM4EALDH1A1CA1CA2POLB
SCHEMBL4851536 0.81 ALDH1A1 (0.44) KDM4EALDH1A1HPGDCA1CA2
Zinc Ion SCHEMBL6913390 0.79 KDM4E (0.47) IKBKBKDM4EALDH1A1HPGDCA1
SCHEMBL6917212 0.79 KDM4E (0.47) IKBKBKDM4EALDH1A1HPGDCA1
SCHEMBL6918561 0.79 KDM4E (0.47) IKBKBKDM4EALDH1A1HPGDCA1
SCHEMBL6914993 0.79 KDM4E (0.47) IKBKBKDM4EALDH1A1HPGDCA1
SCHEMBL6913171 0.79 KDM4E (0.47) IKBKBKDM4EALDH1A1HPGDCA1
SCHEMBL6918557 0.79 KDM4E (0.47) IKBKBKDM4EALDH1A1HPGDCA1
SCHEMBL6908398 0.79 KDM4E (0.47) IKBKBKDM4EALDH1A1HPGDCA1
SCHEMBL6913801 0.79 KDM4E (0.47) IKBKBKDM4EALDH1A1HPGDCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110545854-A method for renal function determination MEDIBEACON INC 2019-12-06 CN disclosed