(Chloromethyl)Benzene

(Chloromethyl)Benzene

SCHEMBL28396267

C=CC(=O)OCCN(C)C.ClCc1ccccc1.O.O.O.O

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of (Chloromethyl)Benzene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 known ✓ P11229 2/20 0.48
THRB known ✓ P10828 1/20 0.48
HRH1 known ✓ P35367 2/20 0.41
CACNA1B known ✓ Q00975 1/20 0.40
CHRM2 known ✓ P08172 1/20 0.39
CHRM3 known ✓ P20309 1/20 0.39
ALDH1A1 P00352 4/20 0.43
TDP1 Q9NUW8 2/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
RECQL P46063 1/20 0.40
APBA1 Q02410 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 2/20 0.39
BCHE P06276 1/20 0.39
LTA4H P09960 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(Chloromethyl)Benzene SCHEMBL169630 0.99 CHRM1 (0.49) CHRM1THRBALDH1A1HRH1TDP1
(Chloromethyl)Benzene SCHEMBL28034643 0.97 CHRM1 (0.48) CHRM1THRBALDH1A1HRH1TDP1
(Chloromethyl)Benzene SCHEMBL30158925 0.90 CHRM1 (0.43) CHRM1THRBALDH1A1HRH1TDP1
(Chloromethyl)Benzene SCHEMBL28529363 0.85 LMNA (0.50) CHRM1THRBALDH1A1POLBSMN1; SMN2
Benzylamine SCHEMBL28520485 0.85 CHRM1 (0.49) CHRM1THRBALDH1A1HRH1TDP1
Hydrochloric Acid SCHEMBL28002276 0.85 CHRM1 (0.49) CHRM1THRBALDH1A1HRH1TDP1
(Chloromethyl)Benzene SCHEMBL8070807 0.85 THRB (0.44) CHRM1THRBALDH1A1TDP1MAPT
SCHEMBL28002275 0.84 CHRM1 (0.46) CHRM1THRBALDH1A1HRH1TDP1
Benzylamine SCHEMBL27761870 0.84 CHRM1 (0.48) CHRM1THRBALDH1A1HRH1TDP1
(Chloromethyl)Benzene SCHEMBL28976987 0.83 THRB (0.43) CHRM1THRBALDH1A1TDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997593-B Method for modifying the rheology of a slurry 埃科莱布美国股份有限公司 2023-01-24 CN disclosed
CN-110997593-A Rheology modifier for slurries 埃科莱布美国股份有限公司 2020-04-10 CN disclosed