SCHEMBL2852748

SCHEMBL2852748

O=C([CH]COC(F)F)NCc1ccsc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.40
SLC1A3 P43003 2/20 0.38
SLC1A2 P43004 2/20 0.38
SLC1A1 P43005 2/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
THRB P10828 1/20 0.38
HPGD P15428 1/20 0.38
TDP1 Q9NUW8 1/20 0.36
LMNA P02545 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
KDM4C Q9H3R0 1/20 0.34
OPRM1 P35372 6/20 0.34
OPRD1 P41143 3/20 0.34
OPRK1 P41145 3/20 0.34
OPRL1 P41146 1/20 0.34
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2851648 0.80 ALDH1A1 (0.51) HPGDLMNA
SCHEMBL2854435 0.79 TSHR (0.48) HPGDLMNA
SCHEMBL2858150 0.78 LMNA (0.52) HPGDLMNA
SCHEMBL2852749 0.77 HPGD (0.43) GRM5SLC1A3SLC1A2SLC1A1HDAC8
SCHEMBL2849991 0.76 RECQL (0.51) HPGDLMNA
SCHEMBL2857248 0.76 CARM1 (0.39)
SCHEMBL18415493 0.75 HDAC6 (0.50) GRM5SLC1A3SLC1A2SLC1A1HDAC8
SCHEMBL2861180 0.74 MMP13 (0.46) HPGDOPRM1
SCHEMBL2856255 0.74 GAA (0.48)
SCHEMBL6668575 0.73 TGM2 (0.56) GRM5HDAC8HDAC6THRBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963277-B1 FLUORINATED COMPOUNDS NPS PHARMA INC (US) 2010-01-20 EP claimed
US-7902401-B2 Fluorinated compounds NPS PHARMACEUTICALS, INC. (US) 2011-03-08 US disclosed
EP-1963277-B1 FLUORINATED COMPOUNDS NPS PHARMA INC (US) 2010-01-20 EP disclosed