SCHEMBL2852353

SCHEMBL2852353

Cc1ccc(C)c(NC(=O)Oc2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.44
MAPT P10636 4/20 0.44
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
RXFP1 Q9HBX9 1/20 0.39
GPR6 P46095 1/20 0.39
MAPK14 Q16539 2/20 0.39
TRPC1 P48995 1/20 0.39
TRPC3 Q13507 1/20 0.39
STIM1 Q13586 1/20 0.39
ORAI1 Q96D31 1/20 0.39
STIM2 Q9P246 1/20 0.39
ACHE P22303 1/20 0.39
CCR1 P32246 1/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850809 0.95 MAPT (0.43) RAB9AMAPTRXFP1MAPK14TRPC1
SCHEMBL2852121 0.92 P2RX7 (0.43) RAB9AMAPTGPR6MAPK14TRPC1
SCHEMBL2853465 0.92 RAB9A (0.44) RAB9AMAPTGPR6TRPC1TRPC3
SCHEMBL2857582 0.92 MAPT (0.42) RAB9AMAPTGPR6TRPC1TRPC3
SCHEMBL2850337 0.91 MAPT (0.40) MAPTCYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL2859508 0.89 CYP1A2 (0.46) RAB9AMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL2858283 0.87 MAPT (0.43) RAB9AMAPTGPR6TRPC1TRPC3
SCHEMBL2853258 0.85 NPY5R (0.45) RAB9AMAPTCYP3A4TRPC1TRPC3
SCHEMBL2854533 0.85 MEN1 (0.46) RAB9AMAPTCYP1A2CYP3A4CYP2C19
SCHEMBL2858515 0.84 MAPT (0.44) MAPTGPR6TRPC1TRPC3STIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed