SCHEMBL2853335

SCHEMBL2853335

COc1ccc(-n2ncc(OC(=O)NCc3ccccc3Cl)c2C)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.48
MAPK8 P45983 1/20 0.48
MAPT P10636 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
P2RX7 Q99572 4/20 0.45
PKM P14618 1/20 0.44
POLB P06746 2/20 0.43
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
GAA P10253 1/20 0.42
THRB P10828 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
RECQL P46063 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2858097 0.91 P2RX7 (0.53) TP53MAPTNPC1RAB9AP2RX7
SCHEMBL2858680 0.90 NPC1 (0.45) TP53MAPK8MAPTSMN1; SMN2NPC1
SCHEMBL2850369 0.89 P2RX7 (0.56) TP53MAPK8MAPTP2RX7PKM
SCHEMBL2857338 0.88 RAB9A (0.47) MAPTSMN1; SMN2NPC1RAB9ANFKB1
SCHEMBL2860234 0.85 HPGD (0.54) TP53MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL2854531 0.84 LMNA (0.52) TP53MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL2856505 0.84 TP53 (0.59) TP53MAPK8MAPTSMN1; SMN2NPC1
SCHEMBL2852417 0.82 MAPT (0.49) TP53MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL2850323 0.82 MAPT (0.47) TP53MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL2856602 0.81 RIPK1 (0.46) TP53MAPTP2RX7MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed