SCHEMBL28536731

SCHEMBL28536731

Nc1cc(OC(F)(F)F)c(-c2ccccc2)c(Cl)c1N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.35
GRIA1 P42261 2/20 0.33
CACNG8 Q8WXS5 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAP2 P11137 1/20 0.32
SCN9A Q15858 3/20 0.32
GRIN2B Q13224 1/20 0.32
KDM4E B2RXH2 2/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
GLA P06280 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28529302 0.80 EPAS1 (0.37) ACLYGRIA1CACNG8ALDH1A1LMNA
SCHEMBL14744335 0.77 GRIA1 (0.39) ACLYGRIA1CACNG8L3MBTL1GRIN2B
SCHEMBL4379379 0.74 L3MBTL1 (0.36) ACLYGRIA1CACNG8L3MBTL1SCN9A
SCHEMBL28535038 0.72 POLB (0.33) L3MBTL1KDM4EALDH1A1LMNAGLA
SCHEMBL28929835 0.69 HSD17B10 (0.46) ACLYL3MBTL1SCN9AKDM4EHSP90AA1
SCHEMBL7396451 0.69 MAPT (0.47) ACLYSCN9AKDM4EHSP90AA1ALDH1A1
SCHEMBL14746409 0.68 RORC (0.40) ACLYGRIA1CACNG8RORCCYP2C9
SCHEMBL14746790 0.67 ALDH1A1 (0.38) L3MBTL1SCN9AKDM4EALDH1A1LMNA
SCHEMBL7937713 0.66 MPL (0.40) GRIA1CACNG8L3MBTL1GRIN2BKDM4E
SCHEMBL31120353 0.66 SCN9A (0.44) L3MBTL1SCN9AKDM4EALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107635970-B Benzimidazolone and benzothiazolone compounds and their use as AMPA receptor modulators 詹森药业有限公司 2021-03-12 CN disclosed