SCHEMBL28779668

SCHEMBL28779668

CCOOCC(C#N)NC(=O)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.49
HDAC1 Q13547 2/20 0.49
HDAC2 Q92769 2/20 0.49
EPHX2 P34913 4/20 0.43
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
TRPV1 Q8NER1 6/20 0.43
NR1H4 Q96RI1 1/20 0.43
TLR7 Q9NYK1 2/20 0.42
RAPGEF3 O95398 1/20 0.40
MCHR1 Q99705 1/20 0.40
POLB P06746 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28545233 0.88 GPR139 (0.48) TRPV1HDAC8
SCHEMBL28566084 0.87 LMNA (0.43) EPHX2PPARGPPARATRPV1
SCHEMBL28550888 0.84 ALDH1A1 (0.48) HDAC3HDAC1HDAC2
SCHEMBL28558833 0.83 L3MBTL1 (0.44) HDAC3HDAC1HDAC2EPHX2NR1H4
SCHEMBL28549384 0.83 MAPT (0.45) HDAC1HDAC6
SCHEMBL28559436 0.82 HTT (0.51) HDAC3HDAC1HDAC2EPHX2POLB
SCHEMBL28554497 0.82 HDAC3 (0.43) HDAC3HDAC1HDAC2POLBHDAC10
SCHEMBL28554447 0.81 CTSL (0.47)
SCHEMBL28557766 0.80 CTSB (0.52) HDAC3HDAC1HDAC2HDAC8
SCHEMBL28550547 0.79 TAS1R3 (0.44) KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112778333-B Tetrahydrooxazolopyridino-azoxanone derivative and application thereof 中国科学院新疆理化技术研究所 2022-07-05 CN disclosed
CN-112724157-B Dihydrooxazolo [5,4-d ] pyrrolo [1,2-a ] pyrimidin-9 (5H) -one derivatives and use thereof 中国科学院新疆理化技术研究所 2022-04-19 CN disclosed
CN-112851692-B Oxazolo [5,4-d ] pyrido [1,2-a ] pyrimidone derivative and application thereof 中国科学院新疆理化技术研究所 2022-04-08 CN disclosed
CN-112851692-A Oxazolo [5,4-d ] pyrido [1,2-a ] pyrimidone derivative and application thereof 中国科学院新疆理化技术研究所 2021-05-28 CN disclosed
CN-112778333-A Tetrahydrooxazolopyridino-azoxanone derivative and application thereof 中国科学院新疆理化技术研究所 2021-05-11 CN disclosed
CN-112724157-A Dihydrooxazolo [5,4-d ] pyrrolo [1,2-a ] pyrimidin-9 (5H) -one derivatives and use thereof 中国科学院新疆理化技术研究所 2021-04-30 CN disclosed