SCHEMBL28801600

SCHEMBL28801600

C=CC(OC(C)=O)c1cc(Br)ccc1F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.34
KAT6A Q92794 1/20 0.34
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
APLNR P35414 2/20 0.32
ACACB O00763 1/20 0.32
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
LMNA P02545 3/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
GAA P10253 1/20 0.31
EGFR P00533 4/20 0.31
KDR P35968 4/20 0.31
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27860279 0.79 APLNR (0.38) DGAT1KAT6AALDH1A1L3MBTL1APLNR
SCHEMBL27628648 0.75 CYP1A2 (0.44) ALDH1A1KMT2AMEN1LMNANPC1
SCHEMBL27913950 0.74 TGM2 (0.39) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL16952185 0.71 LMNA (0.33) DGAT1APLNRLMNA
SCHEMBL9515508 0.71 APLNR (0.48) DGAT1ALDH1A1L3MBTL1APLNRACACB
SCHEMBL933449 0.69 ALDH1A1 (0.33) ALDH1A1KMT2AMEN1LMNAKDM4E
SCHEMBL27697290 0.68 DGAT1 (0.42) DGAT1ALDH1A1L3MBTL1APLNRACACB
SCHEMBL21470340 0.68 MEN1 (0.33) KAT6AAPLNRACACBKMT2AMEN1
SCHEMBL7222153 0.68 HDAC4 (0.43) ALDH1A1KDM4E
SCHEMBL7222151 0.68 HDAC4 (0.43) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958922-A 2,5,6,7-tetrahydro-[1,4]oxazepin-3-ylamine or 2,3,6,7-tetrahydro-[1,4]oxazepin-5-ylamine compounds HOFFMANN LA ROCHE 2013-03-06 CN disclosed