SCHEMBL28819258

SCHEMBL28819258

COc1ccc(C=CC(=O)C=Cc2ccc(OCCN3CCN(S(=O)(=O)c4ccc(C(F)(F)F)cc4)CC3=O)cc2)c(OC)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 4/20 0.45
CYP1B1 Q16678 4/20 0.45
GPR183 P32249 5/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CA2 P00918 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CAPN1 P07384 1/20 0.41
CTSB P07858 1/20 0.41
BACE1 P56817 1/20 0.40
GAA P10253 1/20 0.40
HDAC1 Q13547 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28819259 0.92 GPR183 (0.44) CYP1A1CYP1B1GPR183MEN1MAPT
SCHEMBL28819227 0.86 L3MBTL1 (0.55) CYP1A1CYP1B1GPR183MEN1MAPT
SCHEMBL28819248 0.85 ALDH1A1 (0.43) GPR183MEN1MAPTKMT2ALMNA
SCHEMBL28819260 0.84 PKM (0.53) CYP1A1CYP1B1GPR183MEN1MAPT
SCHEMBL28819245 0.80 LMNA (0.52) GPR183MEN1MAPTKMT2ALMNA
SCHEMBL28819241 0.80 LMNA (0.48) GPR183LMNASMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL28819261 0.76 GPR183 (0.52) GPR183MEN1MAPTKMT2ALMNA
SCHEMBL28819231 0.75 GPR183 (0.62) GPR183LMNAL3MBTL1ALDH1A1
SCHEMBL28819236 0.73 GPR183 (0.62) GPR183MEN1MAPTKMT2ALMNA
SCHEMBL28819256 0.73 PKM (0.67) GPR183MEN1MAPTKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114634465-A Sulfonyl piperazine-containing pentadiene ketone derivative and preparation method and application thereof 贵州大学 2022-06-17 CN disclosed