SCHEMBL28819248

SCHEMBL28819248

COc1ccc(C=CC(=O)C=Cc2ccc(OCCN3CCN(S(=O)(=O)c4cccs4)CC3=O)cc2)c(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.43
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPK1 P28482 2/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
TP53 P04637 1/20 0.43
CYP3A4 P08684 1/20 0.43
CASP1 P29466 1/20 0.43
BRCA1 P38398 1/20 0.43
RECQL P46063 1/20 0.43
CASP7 P55210 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
RAB9A P51151 2/20 0.42
CAPN1 P07384 1/20 0.42
CTSB P07858 1/20 0.42
GPR183 P32249 1/20 0.42
PKM P14618 5/20 0.41
BACE1 P56817 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28819250 0.87 RAB9A (0.54) ALDH1A1KMT2ARAB9AGPR183PKM
SCHEMBL28819258 0.85 CYP1A1 (0.45) ALDH1A1MAPTMEN1KMT2ACAPN1
SCHEMBL28819249 0.83 ALDH1A1 (0.58) ALDH1A1MAPTMEN1KMT2AMAPK1
SCHEMBL28819259 0.83 GPR183 (0.44) ALDH1A1MAPTMEN1KMT2AMAPK1
SCHEMBL28819227 0.71 L3MBTL1 (0.55) ALDH1A1MAPTMEN1KMT2AGPR183
SCHEMBL28838366 0.70 MAPT (0.67) ALDH1A1MAPTMEN1KMT2ARAB9A
SCHEMBL28819245 0.70 LMNA (0.52) ALDH1A1MAPTMEN1KMT2AGPR183
SCHEMBL28819241 0.69 LMNA (0.48) ALDH1A1GPR183PKMLMNASMN1; SMN2
SCHEMBL28819252 0.68 ALDH1A1 (0.76) ALDH1A1KMT2ARAB9AGPR183PKM
SCHEMBL28360809 0.66 CAPN1 (0.85) ALDH1A1MAPTMEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114634465-A Sulfonyl piperazine-containing pentadiene ketone derivative and preparation method and application thereof 贵州大学 2022-06-17 CN disclosed