SCHEMBL28836205

SCHEMBL28836205

CC(C)c1cc(C(=O)NCc2ccccc2)nnc1Nc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.54
MMP13 P45452 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 5/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPT P10636 2/20 0.46
POLB P06746 2/20 0.46
HPGD P15428 5/20 0.46
HSD17B10 Q99714 3/20 0.46
KDM4E B2RXH2 2/20 0.46
LRRK2 Q5S007 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
NPSR1 Q6W5P4 2/20 0.42
GLA P06280 1/20 0.42
EGFR P00533 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28111242 0.90 RAB9A (0.53) SMN1; SMN2MMP13CYP1A2CYP2D6CYP2C19
SCHEMBL28111738 0.76 SMN1; SMN2 (0.48) SMN1; SMN2MMP13CYP1A2CYP2D6CYP2C19
SCHEMBL27021656 0.73 KMT2A (0.65) SMN1; SMN2CYP1A2CYP2C19ALDH1A1MEN1
SCHEMBL28111733 0.73 MMP13 (0.52) SMN1; SMN2MMP13CYP1A2CYP2D6CYP2C19
SCHEMBL5370386 0.69 MMP13 (0.62) SMN1; SMN2MMP13CYP1A2CYP2D6CYP2C19
SCHEMBL17661849 0.69 HPGD (0.60) SMN1; SMN2CYP1A2CYP2C19ALDH1A1MEN1
SCHEMBL21644655 0.67 HSP90AA1 (0.64) SMN1; SMN2CYP2C19ALDH1A1KMT2AHPGD
SCHEMBL2373449 0.66 AMY1A (0.57) SMN1; SMN2MMP13ALDH1A1MEN1KMT2A
SCHEMBL28836629 0.66 VNN1 (0.56) SMN1; SMN2MMP13MEN1KMT2AMAPT
SCHEMBL28111776 0.66 MAPT (0.64) MMP13CYP1A2CYP2C19ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN claimed
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN disclosed