SCHEMBL2888752

SCHEMBL2888752

CCOC(=O)c1cc(-c2ccc(Cl)cc2)n(-c2ccccc2)c1C

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 7/20 0.72
MAPK1 P28482 1/20 0.65
LMNA P02545 2/20 0.60
TP53 P04637 7/20 0.59
MAPT P10636 4/20 0.59
POLB P06746 1/20 0.57
ALDH1A1 P00352 1/20 0.56
HPGD P15428 1/20 0.56
TSHR P16473 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5922342 0.95 CHRNA7 (0.72) CHRNA7MAPK1LMNATP53MAPT
SCHEMBL16403251 0.94 CHRNA7 (0.81) CHRNA7MAPK1LMNATP53MAPT
SCHEMBL5922348 0.91 LMNA (0.69) CHRNA7LMNATP53MAPTPOLB
SCHEMBL7172634 0.89 LMNA (0.67) CHRNA7MAPK1LMNATP53MAPT
SCHEMBL24157321 0.89 CHRNA7 (0.59) CHRNA7MAPK1LMNATP53MAPT
SCHEMBL3027578 0.88 CHRNA7 (0.77) CHRNA7MAPK1LMNAALDH1A1
SCHEMBL2884407 0.88 CHRNA7 (0.72) CHRNA7LMNATP53MAPTPOLB
SCHEMBL19808409 0.87 CHRNA7 (0.74) CHRNA7MAPK1TP53MAPT
SCHEMBL13574377 0.86 CHRNA7 (0.61) CHRNA7MAPK1LMNATP53MAPT
SCHEMBL3025992 0.85 CHRNA7 (0.68) CHRNA7MAPK1LMNATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 137 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240316060-A1 LASER AND BCL-2 INHIBITORS COMBINATION TO TREAT SOLID TUMORS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2024-09-26 US claimed
CN-117186241-A Antibacterial peptide containing LL-37 sequence and application thereof 国科温州研究院(温州生物材料与工程研究所) 2023-12-08 CN claimed
US-20260124276-A1 BIOENGINEERING TERITIARY LYMPHOID STRUCTURES USING CHITOSAN-BASED HYDROGELS H LEE MOFFITT CANCER CENTER AND RESEARCH INST INC (US) 2026-05-07 US disclosed
WO-2026090438-A1 COMPOSITIONS AND METHODS FOR TREATING ACUTE RESPIRATORY DISTRESS SYNDROME DIRECT BIOLOGICS, LLC (US) 2026-04-30 WO disclosed
EP-4728275-A1 METHODS AND ASSAYS FOR IMMUNE PHENOTYPING Immune Functional Diagnostics, LLC (US) 2026-04-22 EP disclosed
EP-4545541-B1 CIRCULARLY POLARIZED LIGHT-EMITTING MATERIAL AND USE, LIGHT-EMITTING DISPLAY DEVICE, AND DISPLAY APPARATUS UNIV ZHEJIANG TECHNOLOGY (CN) 2026-02-18 EP disclosed
US-20260034241-A1 COMPOSITIONS AND METHODS FOR IN VIVO EXPRESSION OF CHIMERIC ANTIGEN RECEPTORS ONCOSENX INC (US) 2026-02-05 US disclosed
US-20260029409-A1 MARKERS FOR DIAGNOSING INFECTIONS MEMED DIAGNOSTICS LTD. (IL) 2026-01-29 US disclosed
US-12485171-B2 Methods of disease activity profiling for personalized therapy management PROMETHEUS LABORATORIES INC. (US) 2025-12-02 US disclosed
US-20250325599-A1 A CLINICAL ISOLATED AVIRULENT STRAIN PROTECTS AGAINST WILDTYPE VIRULENT CLOSTRIDIOIDES DIFFICILE INFECTION THE UNIVERSITY OF CHICAGO (US) 2025-10-23 US disclosed
US-20250305029-A1 GENERATION OF PHASED READ-SETS FOR GENOME ASSEMBLY AND HAPLOTYPE PHASING DOVETAIL GENOMICS, LLC 2025-10-02 US disclosed
EP-3124489-B1 THIAZOLO-PYRIDINE COMPOUNDS AS HIF MODULATORS FIBROGEN INC (US) 2020-07-15 EP disclosed
US-20190106387-A1 NOVEL METHODS, COMPOUNDS, AND COMPOSITIONS FOR ANESTHESIA THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2019-04-11 US disclosed
US-20180022698-A1 NOVEL METHODS, COMPOUNDS, AND COMPOSITIONS FOR ANESTHESIA THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2018-01-25 US disclosed
EP-3124489-A1 THIAZOLO-PYRIDINE COMPOUNDS AS HIF MODULATORS Fibrogen, Inc. (US) 2017-02-01 EP disclosed
EP-2016078-B1 PYRROLO- AND THIAZOLO-PYRIDINE COMPOUNDS AS HIF MODULATORS FIBROGEN INC (US) 2016-06-15 EP disclosed
US-7696223-B2 [(2-bromo-4-hydroxy-1-phenyl-1H-pyrrolo[2,3-c]pyridine-5-carbonyl)-amino]-acetic acid; modulates the stability and/or activity of hypoxia inducible factor (HIF) FIBROGEN, INC. (US) 2010-04-13 US disclosed
EP-2016078-A2 PYRROLO- AND THIAZOLO-PYRIDINE COMPOUNDS AS HIF MODULATORS FIBROGEN, INC. (US) 2009-01-21 EP disclosed
US-20080004309-A1 PYRROLO- AND THIAZOLO-PYRIDINE COMPOUNDS, AND METHODS OF USE THEREOF FIBROGEN, INC. 2008-01-03 US disclosed
WO-2007115315-A2 PYRROLO- AND THIAZOLO-PYRIDINE COMPOUNDS AS HIF MODULATORS FIBROGEN, INC. (US) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180022698-A1 NOVEL METHODS, COMPOUNDS, AND COMPOSITIONS FOR ANESTHESIA GABRA5, GABRA4, GABRA6 CHRNA7 38/4885MAPK1 4520/4885LMNA 3605/4885
US-20260124276-A1 BIOENGINEERING TERITIARY LYMPHOID STRUCTURES USING CHITOSAN-BASED HYDROGELS CCL5, CCR9, CCL11 CHRNA7 2362/4885MAPK1 2777/4885LMNA 4703/4885
US-20260029409-A1 MARKERS FOR DIAGNOSING INFECTIONS AGER, TSG101, ST14 CHRNA7 4733/4885MAPK1 2940/4885LMNA 4267/4885
US-20260034241-A1 COMPOSITIONS AND METHODS FOR IN VIVO EXPRESSION OF CHIMERIC ANTIGEN RECEPTORS CD47, CD74, ICOS CHRNA7 2062/4885MAPK1 4427/4885LMNA 1160/4885
US-20080004309-A1 PYRROLO- AND THIAZOLO-PYRIDINE COMPOUNDS, AND METHODS OF USE THEREOF HIF1AN, HIF1A, EGLN2 CHRNA7 4787/4885MAPK1 3037/4885LMNA 4255/4885
US-20190106387-A1 NOVEL METHODS, COMPOUNDS, AND COMPOSITIONS FOR ANESTHESIA GABRA5, GABRA4, GABRA6 CHRNA7 38/4885MAPK1 4520/4885LMNA 3605/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.