SCHEMBL28912705

SCHEMBL28912705

CC(C)(C)OC(=O)c1cc2cc(NC(=O)CCc3ccccc3O)ccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 2/20 0.46
LEF1 Q9UJU2 1/20 0.44
F11 P03951 2/20 0.43
MMP2 P08253 1/20 0.40
PYGL P06737 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 4/20 0.38
LMNA P02545 2/20 0.38
MAPK1 P28482 1/20 0.38
XDH P47989 1/20 0.38
NPY5R Q15761 1/20 0.37
KDM4E B2RXH2 3/20 0.37
NPC1 O15118 2/20 0.37
ALDH1A1 P00352 2/20 0.37
USP2 O75604 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TP53 P04637 2/20 0.36
POLB P06746 1/20 0.36
MAOA P21397 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24988007 0.87 ALDH1A1 (0.49) MMP13LEF1F11MMP2MAPT
SCHEMBL28941288 0.77 MMP13 (0.62) MMP13MMP2MEN1KMT2AMAPT
SCHEMBL23486667 0.75 MMP13 (0.51) MMP13LEF1F11MMP2KMT2A
SCHEMBL29121378 0.74 MMP13 (0.49) MMP13LEF1MMP2MEN1KMT2A
SCHEMBL28555873 0.73 MMP13 (0.47) MMP13LEF1F11MMP2PYGL
SCHEMBL28555872 0.73 MMP13 (0.47) MMP13LEF1F11MMP2PYGL
SCHEMBL3497422 0.72 EGFR (0.57) MMP13LEF1F11KMT2AKDM4E
SCHEMBL5087408 0.72 LEF1 (0.59) MMP13LEF1PYGLMEN1KMT2A
SCHEMBL6617416 0.72 LEF1 (0.74) MMP13LEF1F11MMP2KMT2A
SCHEMBL7833243 0.71 LEF1 (0.55) MMP13LEF1MMP2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112608303-B Piperazine intermediate, preparation method and application thereof 华南理工大学 2021-10-26 CN disclosed
CN-112608303-A Piperazine intermediate, preparation method and application thereof 华南理工大学 2021-04-06 CN disclosed