SCHEMBL2893669

SCHEMBL2893669

CC(=O)c1cnn(COCC[Si](C)(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.40
ACHE P22303 2/20 0.36
NPC1 O15118 1/20 0.36
KLKB1 P03952 3/20 0.36
DGAT1 O75907 6/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 1/20 0.33
AR P10275 1/20 0.32
MAPT P10636 2/20 0.32
CYP2C19 P33261 1/20 0.32
GFER P55789 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
KLK1 P06870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17723760 0.88 L3MBTL1 (0.54) L3MBTL1ACHENPC1KLKB1
SCHEMBL3698405 0.87 NPC1 (0.46) L3MBTL1ACHENPC1KLKB1DGAT1
SCHEMBL28769640 0.87 L3MBTL1 (0.39) L3MBTL1ACHENPC1KLKB1DGAT1
SCHEMBL20271394 0.85 HPGD (0.39) L3MBTL1ACHENPC1KLKB1DGAT1
SCHEMBL18074418 0.85 L3MBTL1 (0.41) L3MBTL1ACHENPC1KLKB1DGAT1
SCHEMBL31196012 0.84 KLKB1 (0.40) L3MBTL1ACHENPC1KLKB1LMNA
SCHEMBL31639060 0.84 L3MBTL1 (0.37) L3MBTL1ACHENPC1KLKB1DGAT1
SCHEMBL27166661 0.84 L3MBTL1 (0.37) L3MBTL1ACHENPC1KLKB1DGAT1
SCHEMBL16881589 0.83 ACHE (0.57) L3MBTL1ACHENPC1KLKB1DGAT1
SCHEMBL17723736 0.83 L3MBTL1 (0.39) L3MBTL1KLKB1DGAT1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4734985-A1 PREVENTION, INHIBITION OR TREATMENT OF CONDITIONS OR DISORDERS MEDIATED BY UROCANATE REDUCTASE IMPLEXION PHARMA AB (SE) 2026-05-06 EP disclosed
US-20260116881-A1 KIF MODULATOR COMPOUNDS AND METHODS OF USE IAMBIC THERAPEUTICS INC (US) 2026-04-30 US disclosed
WO-2025136936-A1 AGONISTS OF TREM2 ACTIVITY MERCK SHARP & DOHME LLC (US) 2025-06-26 WO disclosed
WO-2025003469-A1 PREVENTION, INHIBITION OR TREATMENT OF CONDITIONS OR DISORDERS MEDIATED BY UROCANATE REDUCTASE IMPLEXION PHARMA AB (SE) 2025-01-02 WO disclosed
US-20240101531-A1 PYRIDINAMINE DERIVATIVES AND THEIR USE AS POTASSIUM CHANNEL MODULATORS XENON PHARMACEUTICALS INC. (CA) 2024-03-28 US disclosed
WO-2023239729-A1 PYRIDINAMINE DERIVATIVES AND THEIR USE AS POTASSIUM CHANNEL MODULATORS XENON PHARMACEUTICALS INC. (CA) 2023-12-14 WO disclosed
EP-3356360-A1 THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF Genentech, Inc. (US) 2018-08-08 EP disclosed
US-10010539-B2 Pyrazole, triazole and tetrazole orexin receptor antagonists MERCK SHARP & DOHME CORP. (US) 2018-07-03 US disclosed
US-10010539-B2 Pyrazole, triazole and tetrazole orexin receptor antagonists MERCK SHARP & DOHME CORP. (US) 2018-07-03 US disclosed
EP-3271353-A1 3-(4-ETHYNYLPHENYL)HEXAHYDROPYRIMIDIN-2,4-DIONE DERIVATIVES AS MODULATORS OF MGLUR4 F. Hoffmann-La Roche AG (CH) 2018-01-24 EP disclosed
US-20170319560-A1 PYRAZOLE, TRIAZOLE AND TETRAZOLE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2017-11-09 US disclosed
WO-2016146600-A1 3-(4-ETHYNYLPHENYL)HEXAHYDROPYRIMIDIN-2,4-DIONE DERIVATIVES AS MODULATORS OF MGLUR4 F. HOFFMANN-LA ROCHE AG (CH) 2016-09-22 WO disclosed
WO-2016065586-A1 PYRAZOLE, TRIAZOLE AND TETRAZOLE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-05-06 WO disclosed
US-8440666-B2 Pyridazinone compounds and P2X7 receptor inhibitors NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2013-05-14 US disclosed
US-8440666-B2 Pyridazinone compounds and P2X7 receptor inhibitors NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2013-05-14 US disclosed
US-8440666-B2 Pyridazinone compounds and P2X7 receptor inhibitors NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2013-05-14 US disclosed
US-20100286390-A1 PYRIDAZINONE COMPOUNDS AND P2X7 RECEPTOR INHIBITORS NISSAN CHEMICAL INDUSTRIES LIMITED 2010-11-11 US disclosed
US-20100286390-A1 PYRIDAZINONE COMPOUNDS AND P2X7 RECEPTOR INHIBITORS NISSAN CHEMICAL INDUSTRIES LIMITED 2010-11-11 US disclosed
EP-2203429-A1 PYRIDAZINONE DERIVATIVES AND USE THEREOF AS P2X7 RECEPTOR INHIBITORS Nissan Chemical Industries, Ltd. (JP) 2010-07-07 EP disclosed
WO-2009057827-A1 PYRIDAZINONE DERIVATIVES AND USE THEREOF AS P2X7 RECEPTOR INHIBITORS NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2009-05-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260116881-A1 KIF MODULATOR COMPOUNDS AND METHODS OF USE KIF2C, KIF5B, KIF5C L3MBTL1 3279/4885ACHE 4567/4885NPC1 107/4885
US-10010539-B2 Pyrazole, triazole and tetrazole orexin receptor antagonists HCRTR2, HCRTR1, NPY5R L3MBTL1 4767/4885ACHE 2101/4885NPC1 1434/4885
US-20240101531-A1 PYRIDINAMINE DERIVATIVES AND THEIR USE AS POTASSIUM CHANNEL MODULATORS KCNA1, KCNB1, KCNB2 L3MBTL1 2240/4885ACHE 343/4885NPC1 1618/4885
US-20100286390-A1 PYRIDAZINONE COMPOUNDS AND P2X7 RECEPTOR INHIBITORS P2RY1, P2RX7, P2RX1 L3MBTL1 4862/4885ACHE 3033/4885NPC1 1850/4885
US-20170319560-A1 PYRAZOLE, TRIAZOLE AND TETRAZOLE OREXIN RECEPTOR ANTAGONISTS HCRTR2, HCRTR1, NPY5R L3MBTL1 4621/4885ACHE 2086/4885NPC1 1438/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.