Tromethamine

Tromethamine

SCHEMBL2898170

CC(=O)O.CNCO.NC(CO)(CO)CO

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DHFRGARTPTGFRPTGIRPTGS1PTGS2TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8envmurAthyA

The experimentally established mechanism targets of Tromethamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
KMT2A Q03164 1/20 0.48
FFAR3 O14843 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tromethamine SCHEMBL466420 0.87 MEN1 (0.62) MEN1LMNAKMT2A
Tromethamine SCHEMBL4581519 0.87 LMNA (0.62) MEN1LMNAKMT2AFFAR3LCK
Tromethamine SCHEMBL7347818 0.87 LMNA (0.62) MEN1LMNAKMT2AFFAR3LCK
Tromethamine SCHEMBL194002 0.87 LMNA (0.62) MEN1LMNAKMT2AFFAR3LCK
Tromethamine SCHEMBL8530527 0.85 MEN1 (0.59) MEN1LMNAKMT2A
Tromethamine SCHEMBL8573552 0.85 MEN1 (0.59) MEN1LMNAKMT2A
Acetic Acid SCHEMBL3431821 0.82 FFAR3 (0.50) LMNAFFAR3LCKFYN
Acetic Acid SCHEMBL31396472 0.82
Tromethamine SCHEMBL5891164 0.80 MEN1 (0.53) MEN1LMNAKMT2AFFAR3LCK
Tromethamine SCHEMBL3473649 0.80 LMNA (0.53) MEN1LMNAKMT2AFFAR3LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432221-B1 ONE-STEP IN SITU HYBRIDIZATION ASSAY APROGENEX INC (US) 1997-05-28 EP claimed
US-9164099-B2 Site-specific labeling of affinity tags in fusion proteins Life Technologies Corporation (US) 2015-10-20 US disclosed
US-20140038856-A1 Site-specific labeling of affinity tags in fusion proteins Life Technologies Corporation (US) 2014-02-06 US disclosed
US-20120270757-A1 SITE-SPECIFIC LABELING OF AFFINITY TAGS IN FUSION PROTEINS Life Technologies Corporation (US) 2012-10-25 US disclosed
EP-2217608-B1 PHOTOLUMINESCENT METAL COMPLEXES FOR PROTEIN STAINING BIO RAD LABORATORIES (US) 2012-09-05 EP disclosed
EP-2217608-A1 PHOTOLUMINESCENT METAL COMPLEXES FOR PROTEIN STAINING Bio-Rad Laboratories, Inc. (US) 2010-08-18 EP disclosed
EP-2089429-A2 PROCESS FOR PREPARING UNAGGREGATED ANTIBODY FC DOMAINS Centocor Ortho Biotech Inc. (US) 2009-08-19 EP disclosed
WO-2009067603-A1 PHOTOLUMINESCENT METAL COMPLEXES FOR PROTEIN STAINING BIO-RAD LABORATORIES, INC. (US) 2009-05-28 WO disclosed
US-20090131640-A1 PHOTOLUMINESCENT METAL COMPLEXES FOR PROTEIN STAINING BIO-RAD LABORATORIES, INC. (US) 2009-05-21 US disclosed
US-20090081722-A1 SITE-SPECIFIC LABELING OF AFFINITY TAGS IN FUSION PROTEINS INVITROGEN CORPORATION (US) 2009-03-26 US disclosed
US-20060141554-A1 Site-specific labeling of affinity tags in fusion proteins INVITROGEN CORP. 2006-06-29 US disclosed
US-20050233307-A1 Site-specific labeling of affinity tags in fusion proteins Life Technologies Corporation 2005-10-20 US disclosed
WO-2005083394-A2 METHODS FOR DETECTING ANIONIC AND NON-ANIONIC PROTEINS USING CARBOCYANINE DYES MOLECULAR PROBES, INC. (US) 2005-09-09 WO disclosed
EP-1546359-A2 SITE-SPECIFIC LABELING OF AFFINITY TAGS IN FUSION PROTEINS Molecular Probes Inc. (US) 2005-06-29 EP disclosed
WO-2005038460-A2 SITE-SPECIFIC LABELING OF AFFINITY TAGS IN FUSION PROTEINS MOLECULAR PROBES, INC. (US) 2005-04-28 WO disclosed
WO-2004025259-A2 SITE-SPECIFIC LABELING OF AFFINITY TAGS IN FUSION PROTEINS MOLECULAR PROBES, INC. (US) 2004-03-25 WO disclosed
US-6316267-B1 COMBINING SAMPLE MIXTURE CONTAININGPOLY(AMINO ACID) WITH A STAINING MIXTURE THAT CONTAINS ONE OR MORE METAL COMPLEXES; INCUBATING COMBINED MIXTURE; ILLUMINATING SAID DYE-POLY(AMINO ACID) COMPLEX; OBSERVING DETECTABLE OPTICAL RESPONSE MOLECULAR PROBES, INC. 2001-11-13 US disclosed
EP-1042676-A1 LUMINESCENT PROTEIN STAINS CONTAINING TRANSITION METAL COMPLEXES Molecular Probes Inc. (US) 2000-10-11 EP disclosed
WO-2000025139-A1 LUMINESCENT PROTEIN STAINS CONTAINING TRANSITION METAL COMPLEXES MOLECULAR PROBES, INC. (US) 2000-05-04 WO disclosed
US-4205130-A AFFINITY VHROMATORGAPHY, ISOELECTRIC FOCUSING VIHKO PIRKKO 1980-05-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060141554-A1 Site-specific labeling of affinity tags in fusion proteins APBA1, F13A1, F13B MEN1 320/4885LMNA 114/4885KMT2A 1830/4885
US-20090131640-A1 PHOTOLUMINESCENT METAL COMPLEXES FOR PROTEIN STAINING NR2E3, NR2C2, ORC3 MEN1 4674/4885LMNA 4298/4885KMT2A 3006/4885
US-20120270757-A1 SITE-SPECIFIC LABELING OF AFFINITY TAGS IN FUSION PROTEINS APBA1, NAPA, F13B MEN1 271/4885LMNA 115/4885KMT2A 1632/4885
US-20090081722-A1 SITE-SPECIFIC LABELING OF AFFINITY TAGS IN FUSION PROTEINS APBA1, F13A1, F13B MEN1 320/4885LMNA 114/4885KMT2A 1830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.