SCHEMBL29138623

SCHEMBL29138623

C[C@H]1CC(c2ncc(Cl)cn2)CCN1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.44
HCRTR1 O43613 4/20 0.35
HCRTR2 O43614 3/20 0.35
BRD4 O60885 1/20 0.34
CCL2 P13500 1/20 0.34
BRD2 P25440 1/20 0.34
EP300 Q09472 1/20 0.34
BRD3 Q15059 1/20 0.34
BRDT Q58F21 1/20 0.34
CREBBP Q92793 1/20 0.34
AOC3 Q16853 1/20 0.34
SMO Q99835 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
SMYD3 Q9H7B4 2/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
ROCK2 O75116 4/20 0.33
PRKG1 Q13976 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29138594 0.83 HCRTR2 (0.36) HSD11B1HCRTR1HCRTR2SMYD3ROCK2
SCHEMBL29138621 0.82 GPR119 (0.44) HSD11B1
SCHEMBL30639338 0.82 GPR119 (0.44) HSD11B1
SCHEMBL3950691 0.77 DRD2 (0.44) HSD11B1
SCHEMBL2636853 0.74 HSD11B1 (0.60) HSD11B1AOC3
SCHEMBL27195383 0.71 CCNE1 (0.34) SMYD3ROCK2PRKG1
SCHEMBL25189423 0.70 TRPC6 (0.43)
SCHEMBL17667436 0.70 ROCK2 (0.44) HSD11B1ROCK2PRKG1
SCHEMBL15646781 0.69 HSD11B1 (0.38) HSD11B1HCRTR2SMOSMYD3CHRM2
SCHEMBL1740550 0.69 HSD11B1 (0.48) HSD11B1AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117247395-A PDE4B inhibitors 武汉人福创新药物研发中心有限公司 2023-12-19 CN disclosed