SCHEMBL2921165

SCHEMBL2921165

O=C(O)Oc1ccnc(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 4/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM1A O60341 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
AR P10275 5/20 0.37
KMT2A Q03164 2/20 0.33
MAPT P10636 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
KDM6B O15054 1/20 0.33
TET3 O43151 1/20 0.33
KDM4A O75164 1/20 0.33
BBOX1 O75936 1/20 0.33
KDM5A P29375 1/20 0.33
KDM5C P41229 1/20 0.33
ASPH Q12797 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25348842 0.87 LMNA (0.46) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL18641430 0.83 KMT2A (0.52) ALDH1A1KDM4ESMN1; SMN2KDM1AHDAC1
SCHEMBL2637576 0.80 CCR1 (0.52) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL27529858 0.79 ACHE (0.46) ALDH1A1KDM4ESMN1; SMN2ARKMT2A
SCHEMBL15819754 0.79 ELANE (0.49) AR
Hydrochloric Acid SCHEMBL6850653 0.78 CCR1 (0.50) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL246279 0.78 LOXL2 (0.36) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL8302350 0.78 ALOX15 (0.50) ALDH1A1KDM4ESMN1; SMN2KMT2AMAPT
SCHEMBL9566767 0.78 NOS3 (0.38) KDM4EMAPTKDM5AKDM4CKDM5B
SCHEMBL753937 0.78 LOX (0.43) ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225223-B1 ORGANIC COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2017-01-11 EP disclosed
EP-2205590-B1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2014-06-04 EP disclosed
EP-2251338-A2 Organic compounds Boehringer Ingelheim International GmbH (DE) 2010-11-17 EP disclosed
EP-2225223-A2 ORGANIC COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-09-08 EP disclosed
EP-2205590-A1 CGRP ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2010-07-14 EP disclosed
WO-2009065919-A2 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-05-28 WO disclosed
WO-2009050232-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed