SCHEMBL2930742

SCHEMBL2930742

Cc1cccc(C(=O)N2C[C@H]3C[C@H]3[C@H]2C(N)=O)c1-c1cncnc1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.35
PIK3CD O00329 1/20 0.34
CYP46A1 Q9Y6A2 1/20 0.34
HCRTR2 O43614 8/20 0.34
ALDH1A1 P00352 1/20 0.34
HCRTR1 O43613 12/20 0.34
PKN1 Q16512 1/20 0.32
PKN2 Q16513 1/20 0.32
PRCP P42785 1/20 0.32
GRM5 P41594 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2932492 0.89 MKNK1 (0.40) PIK3CAPIK3CDCYP46A1HCRTR2ALDH1A1
SCHEMBL2924242 0.86 FABP4 (0.42) PIK3CAPIK3CDCYP46A1HCRTR2ALDH1A1
SCHEMBL2930954 0.85 POLB (0.39) PIK3CAPIK3CDCYP46A1HCRTR2ALDH1A1
SCHEMBL2930744 0.85 HCRTR2 (0.37) PIK3CDCYP46A1HCRTR2HCRTR1PRCP
SCHEMBL2931912 0.83 APOB (0.38) PIK3CDHCRTR2ALDH1A1HCRTR1
SCHEMBL2931039 0.82 HCRTR2 (0.39) PIK3CDHCRTR2HCRTR1GRM5
SCHEMBL2930073 0.82 PDE4B (0.37) HCRTR2HCRTR1GRM5
SCHEMBL2928147 0.81 HCRTR1 (0.36) PIK3CAPIK3CDHCRTR2ALDH1A1HCRTR1
SCHEMBL2926433 0.81 MGLL (0.38) PIK3CAPIK3CDHCRTR2ALDH1A1HCRTR1
SCHEMBL2925490 0.80 PIK3CD (0.37) PIK3CDHCRTR2ALDH1A1HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed