SCHEMBL2930744

SCHEMBL2930744

Cc1cccc(C(=O)N2C[C@H]3C[C@H]3[C@H]2CN)c1-c1cncnc1

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 14/20 0.37
HCRTR1 O43613 16/20 0.36
CYP46A1 Q9Y6A2 1/20 0.35
PIK3CD O00329 1/20 0.33
PRCP P42785 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2932494 0.90 HCRTR2 (0.38) HCRTR2HCRTR1CYP46A1
SCHEMBL2924244 0.87 CYP46A1 (0.39) HCRTR2HCRTR1CYP46A1PIK3CDPRCP
SCHEMBL2930955 0.86 HCRTR2 (0.38) HCRTR2HCRTR1CYP46A1PIK3CDPRCP
SCHEMBL2930742 0.85 PIK3CA (0.35) HCRTR2HCRTR1CYP46A1PIK3CDPRCP
SCHEMBL2931914 0.85 HCRTR2 (0.39) HCRTR2HCRTR1CYP46A1PIK3CD
SCHEMBL2931040 0.82 HCRTR2 (0.40) HCRTR2HCRTR1PIK3CD
SCHEMBL2930074 0.82 SLC6A7 (0.35) HCRTR2HCRTR1
SCHEMBL2928151 0.82 HCRTR2 (0.35) HCRTR2HCRTR1
SCHEMBL2933639 0.81 PAX8 (0.39) PRCP
SCHEMBL2926435 0.80 MGLL (0.37) HCRTR2HCRTR1PIK3CDPRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed