SCHEMBL29375416

SCHEMBL29375416

Brc1cncc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCZ Q05513 1/20 0.46
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
ADRA1A P35348 1/20 0.44
KDM4E B2RXH2 2/20 0.41
GPR3 P46089 1/20 0.41
CYP11B2 P19099 9/20 0.39
CYP11B1 P15538 8/20 0.39
CYP3A4 P08684 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HSD17B10 Q99714 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
LMNA P02545 2/20 0.38
CYP2A6 P11509 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL111247 1.00 PRKCZ (0.46) PRKCZADRA2AADRA2BADRA2CADRA1A
Iodide SCHEMBL27879062 0.98 PRKCZ (0.44) PRKCZADRA2AADRA2BADRA2CADRA1A
SCHEMBL27680594 0.90 PRKCZ (0.40) PRKCZADRA2AADRA2BADRA2CADRA1A
SCHEMBL9871846 0.82 CYP3A4 (0.46) PRKCZADRA2AADRA2BADRA2CADRA1A
SCHEMBL4068814 0.80 HASPIN (0.39) PRKCZADRA2AADRA2BADRA2CADRA1A
SCHEMBL12441263 0.76 IMPDH2 (0.48) ADRA2AADRA2BADRA2CADRA1AKDM4E
SCHEMBL20873066 0.75 PRKCZ (0.64) PRKCZADRA2AADRA2BADRA2CADRA1A
SCHEMBL19656321 0.74 IMPDH2 (0.47) PRKCZADRA2AADRA2BADRA2CADRA1A
SCHEMBL29862478 0.74 IMPDH2 (0.47) PRKCZADRA2AADRA2BADRA2CADRA1A
SCHEMBL6993140 0.74 CYP11B1 (0.44) PRKCZKDM4ECYP11B2CYP11B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12202816-B2 Compounds as NADPH oxidase inhibitors CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2025-01-21 US disclosed
EP-4081299-B1 DIHYDRO-CYCLOPENTA-ISOQUINOLINE DERIVATIVES UCB Biopharma SRL (BE) 2024-09-25 EP disclosed
EP-4333819-A1 TREATMENT OF PHARMACORESISTANT EPILEPSY Katholieke Universiteit Leuven (BE) 2024-03-13 EP disclosed
US-20230192646-A1 DIHYDRO-CYCLOPENTA-ISOQUINOLINE DERIVATIVES UCB Biopharma SRL (BE) 2023-06-22 US disclosed
WO-2023081452-A1 SMALL-MOLECULE DEGRADERS OF CDK8 AND CDK19 UNIVERSITY OF SOUTH CAROLINA (US) 2023-05-11 WO disclosed
WO-2022233877-A1 TREATMENT OF PHARMACORESISTANT EPILEPSY KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-11-10 WO disclosed
EP-4081299-A1 DIHYDRO-CYCLOPENTA-ISOQUINOLINE DERIVATIVES UCB Biopharma SRL (BE) 2022-11-02 EP disclosed
US-11479546-B2 Antimalarial hexahydropyrimidine analogues UCB Biopharma SRL 2022-10-25 US disclosed
US-20220033379-A1 NOVEL COMPOUNDS AS NADPH OXIDASE INHIBITORS CALLIDITAS THERAPEUTICS SUISSE SA (CH) 2022-02-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11479546-B2 Antimalarial hexahydropyrimidine analogues G6PD, DPYD, DHODH PRKCZ 4030/4885ADRA2A 2928/4885ADRA2B 2728/4885
US-12202816-B2 Compounds as NADPH oxidase inhibitors CYBB, NOX1, NOX4 PRKCZ 1087/4885ADRA2A 2520/4885ADRA2B 1773/4885
US-20230192646-A1 DIHYDRO-CYCLOPENTA-ISOQUINOLINE DERIVATIVES FCER2, FCGR2A, FCGR1A PRKCZ 539/4885ADRA2A 302/4885ADRA2B 343/4885
US-20220033379-A1 NOVEL COMPOUNDS AS NADPH OXIDASE INHIBITORS CYBB, NOX1, NOX4 PRKCZ 935/4885ADRA2A 2422/4885ADRA2B 1555/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.