Camostat

Camostat

SCHEMBL29376746

CN(C)C(=O)COC(=O)Cc1ccc(OC(=O)c2ccc(N=C(N)N)cc2)cc1.CS(=O)(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of Camostat. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 known ✓ P00734 5/20 1.00
ADRA1A known ✓ P35348 1/20 0.90
PRSS1 P07477 12/20 1.00
KLK1 P06870 4/20 1.00
PRSS2 P07478 4/20 0.90
PRSS3 P35030 4/20 0.90
HGFAC Q04756 3/20 0.90
TMPRSS2 O15393 2/20 0.90
SLC22A2 O15244 1/20 0.90
HPN P05981 1/20 0.90
CTSL P07711 1/20 0.90
CNR1 P21554 1/20 0.90
OPRD1 P41143 1/20 0.90
KCNH2 Q12809 1/20 0.90
SLC47A2 Q86VL8 1/20 0.90
SLC47A1 Q96FL8 1/20 0.90
ACR P10323 7/20 0.61
TMPRSS15 P98073 3/20 0.58
FTO Q9C0B1 1/20 0.52
PLG P00747 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Camostat SCHEMBL125270 0.95 PRSS1 (1.00) PRSS1F2KLK1PRSS2PRSS3
Camostat SCHEMBL871583 0.83 PRSS1 (0.72) PRSS1F2KLK1PRSS2PRSS3
SCHEMBL15571972 0.83 PRSS1 (0.70) PRSS1F2KLK1PRSS2PRSS3
SCHEMBL1649708 0.82 PRSS1 (1.00) PRSS1F2KLK1PRSS2PRSS3
SCHEMBL21920058 0.81 PRSS1 (0.74) PRSS1F2KLK1PRSS2PRSS3
SCHEMBL4752946 0.79 PRSS1 (0.66) PRSS1F2KLK1PRSS2PRSS3
SCHEMBL20008640 0.79 PRSS1 (0.68) PRSS1F2KLK1PRSS2PRSS3
Camostat SCHEMBL125269 0.79 PRSS1 (0.68) PRSS1F2KLK1PRSS2PRSS3
SCHEMBL13283061 0.79 PRSS1 (0.68) PRSS1F2KLK1PRSS2PRSS3
Camostat SCHEMBL2782237 0.78 PRSS1 (0.67) PRSS1F2KLK1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
EP-4680248-A1 PRODUCTS OF MANUFACTURE AND THERAPEUTIC COMPOSITIONS FOR TREATING, AMELIORATING OR PREVENTING VIRAL INFECTIONS AND METHODS FOR MAKING AND USING THEM Topelia Aust Limited (ACN 652 771 670) (AU) 2026-01-21 EP claimed
WO-2024187239-A1 PRODUCTS OF MANUFACTURE AND THERAPEUTIC COMPOSITIONS FOR TREATING, AMELIORATING OR PREVENTING VIRAL INFECTIONS AND METHODS FOR MAKING AND USING THEM TOPELIA AUST LIMITED (ACN 652 771 670) (AU) 2024-09-19 WO claimed
EP-4189397-A2 METHODS FOR THE DETERMINATION OF THE PREDISPOSITION FOR A SEVERE OR CRITICAL COURSE OF A COVID-19-DISEASE FROM A MILD OR MODERATE COURSE OF A COVID-19-DISEASE IN A SUBJECT Sciomics GmbH (DE) 2023-06-07 EP claimed
CN-116194114-A Cathepsin inhibitors for preventing or treating viral infections 葛兰素史密斯克莱知识产权发展有限公司 2023-05-30 CN claimed
US-20230158259-A1 PRODUCTS OF MANUFACTURE AND METHODS FOR TREATING, AMELIORATING OR PREVENTING MICROBIAL INFECTIONS TOPELIA AUST LIMITED (652 771 670) (AU) 2023-05-25 US claimed
CN-115955965-A Products of manufacture and methods for treating, ameliorating or preventing microbial infections 拓比利亚欧斯特有限公司 2023-04-11 CN claimed
EP-4138832-A1 PRODUCTS OF MANUFACTURE AND METHODS FOR TREATING, AMELIORATING OR PREVENTING MICROBIAL INFECTIONS Topelia Aust Limited (AU) 2023-03-01 EP claimed
EP-4125919-A1 CATHEPSIN INHIBITORS FOR PREVENTING OR TREATING VIRAL INFECTIONS GlaxoSmithKline Intellectual Property Development Limited (GB) 2023-02-08 EP claimed
WO-2022028917-A2 METHODS FOR THE DETERMINATION OF THE PREDISPOSITION FOR A SEVERE OR CRITICAL COURSE OF A COVID-19-DISEASE FROM A MILD OR MODERATE COURSE OF A COVID-19-DISEASE IN A SUBJECT SCIOMICS GMBH (DE) 2022-02-10 WO claimed
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US disclosed
EP-4680248-A1 PRODUCTS OF MANUFACTURE AND THERAPEUTIC COMPOSITIONS FOR TREATING, AMELIORATING OR PREVENTING VIRAL INFECTIONS AND METHODS FOR MAKING AND USING THEM Topelia Aust Limited (ACN 652 771 670) (AU) 2026-01-21 EP disclosed
US-12502381-B2 Serine protease inhibitor for treating coronavirus infection REDHILL BIOPHARMA LTD. (IL) 2025-12-23 US disclosed
CN-117695284-B Treatment of coronavirus infection 红山生物医药有限公司 2025-06-17 CN disclosed
US-20250188022-A1 PROCESS FOR THE PREPARATION OF NAFAMOSTAT, CAMOSTAT AND THEIR DERIVATIVES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2025-06-12 US disclosed
WO-2022066823-A1 CORONAVIRUS REPLICONS FOR ANTIVIRAL SCREENING AND TESTING MERCK SHARP & DOHME CORP. (US) 2022-03-31 WO disclosed
US-11278602-B2 Medicine for Covid-19 and treatment Therapeutica Borealis Oy (FI) 2022-03-22 US disclosed
WO-2022049177-A1 ANTIVIRAL PHARMACEUTICAL COMPOSITION FOR TOPICAL ADMINISTRATION CHRISTIAN-ALBRECHTS-UNIVERSITÄT ZU KIEL (DE) 2022-03-10 WO disclosed
EP-3964207-A1 ANTIVIRAL PHARMACEUTICAL COMPOSITION FOR TOPICAL ADMINISTRATION Christian-Albrechts-Universität zu Kiel (DE) 2022-03-09 EP disclosed
WO-2022028917-A2 METHODS FOR THE DETERMINATION OF THE PREDISPOSITION FOR A SEVERE OR CRITICAL COURSE OF A COVID-19-DISEASE FROM A MILD OR MODERATE COURSE OF A COVID-19-DISEASE IN A SUBJECT SCIOMICS GMBH (DE) 2022-02-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250188022-A1 PROCESS FOR THE PREPARATION OF NAFAMOSTAT, CAMOSTAT AND THEIR DERIVATIVES TPMT, ADH1C, ADH1A F2 1213/4885ADRA1A 3293/4885PRSS1 1209/4885
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS ACE, MAVS, SARS1 F2 828/4885ADRA1A 2150/4885PRSS1 281/4885
US-12502381-B2 Serine protease inhibitor for treating coronavirus infection PRSS1, ACE, TMPRSS2 F2 129/4885ADRA1A 3326/4885PRSS1 1/4885
US-11278602-B2 Medicine for Covid-19 and treatment ACE2, HAVCR2, TMPRSS2 F2 2277/4885ADRA1A 2039/4885PRSS1 148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.