SCHEMBL29645745

SCHEMBL29645745

O=c1nccccc1Nc1nc2c(C(F)(F)F)cccc2c2nc(-c3cc[nH]n3)nn12

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
P2RX7 Q99572 9/20 0.33
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
RET P07949 1/20 0.32
CCNB1 P14635 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
SCN9A Q15858 3/20 0.31
PARP1 P09874 1/20 0.31
SLC40A1 Q9NP59 1/20 0.31
SLC11A2 P49281 1/20 0.31
DHODH Q02127 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29645738 0.86 NTRK1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL29645837 0.84 EGFR (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL29645786 0.84 MAPT (0.42)
SCHEMBL29646148 0.83 LMNA (0.39) SCN9A
SCHEMBL29645682 0.83 ADORA3 (0.40) P2RX7
SCHEMBL29645803 0.83 POLB (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL29645914 0.82 NR1H2 (0.40) P2RX7
SCHEMBL29646083 0.81 MAPT (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL29645597 0.80 TRPA1 (0.34) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL29646123 0.79 P2RX7 (0.33) P2RX7DHODHHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN claimed