SCHEMBL29689092

SCHEMBL29689092

O=C(O)c1cc2ncccc2o1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.49
CSNK2A1 P68400 3/20 0.49
CSNK2A2 P19784 2/20 0.49
CSNK2B P67870 2/20 0.49
CSNK2A3 Q8NEV1 2/20 0.49
USP2 O75604 1/20 0.49
PTGS1 P23219 1/20 0.49
PIM1 P11309 5/20 0.46
PIM2 Q9P1W9 2/20 0.46
CHRNB2 P17787 1/20 0.44
CHRNA4 P43681 1/20 0.44
TDP1 Q9NUW8 4/20 0.42
L3MBTL1 Q9Y468 3/20 0.42
HSD17B10 Q99714 2/20 0.42
MAPT P10636 2/20 0.42
TSHR P16473 2/20 0.42
GLA P06280 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
NAPRT Q6XQN6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4128614 1.00 KDM4E (0.49) KDM4ECSNK2A1CSNK2A2CSNK2BCSNK2A3
SCHEMBL29686936 0.86 CHRNB2 (0.44) KDM4ECHRNB2CHRNA4MAPTNPC1
SCHEMBL17749939 0.84 ALDH1A1 (0.44) KDM4ECHRNB2CHRNA4L3MBTL1HSD17B10
SCHEMBL6281582 0.80 HTT (0.50) KDM4ECHRNB2CHRNA4TDP1L3MBTL1
SCHEMBL11248491 0.78 GPR35 (0.57) KDM4ECHRNB2CHRNA4TDP1L3MBTL1
SCHEMBL24776512 0.78 MEN1 (0.40) USP2CHRNB2CHRNA4HSD17B10MAPT
SCHEMBL24620866 0.77 F7 (0.46) KDM4EUSP2PIM1PIM2L3MBTL1
SCHEMBL30973431 0.75 PIM1 (0.42) KDM4ECSNK2A1CSNK2A2CSNK2BCSNK2A3
SCHEMBL31429009 0.75 RAB9A (0.52) KDM4EL3MBTL1HSD17B10MAPTHPGD
SCHEMBL10513311 0.74 CA2 (0.54) CHRNB2CHRNA4HPGDHTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118324772-A Synthesis method and intermediate of furan [3,2-b ] pyridine derivative 北京颖诺凯胜科技有限公司 2024-07-12 CN claimed
EP-3856179-B1 MONOACYLGLYCEROL LIPASE MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2026-05-13 EP disclosed
CN-113164459-B Monoacylglycerol lipase modulators 詹森药业有限公司 2024-09-03 CN disclosed
CN-118324772-A Synthesis method and intermediate of furan [3,2-b ] pyridine derivative 北京颖诺凯胜科技有限公司 2024-07-12 CN disclosed
CN-118324772-A Synthesis method and intermediate of furan [3,2-b ] pyridine derivative 北京颖诺凯胜科技有限公司 2024-07-12 CN disclosed
US-11993601-B2 Monoacylglycerol lipase modulators JANSSEN PHARMACEUTICA NV 2024-05-28 US disclosed
US-20230242531-A1 Monoacylglycerol Lipase Modulators JANSSEN PHARMACEUTICA NV (BE) 2023-08-03 US disclosed
US-11597728-B2 Monoacylglycerol lipase modulators JANSSEN PHARMACEUTICA NV (BE) 2023-03-07 US disclosed
US-20220315583-A1 Monoacylglycerol Lipase Modulators JANSSEN PHARMACEUTICA NV (BE) 2022-10-06 US disclosed
EP-4007758-A1 BIS-[N-((5-CARBAMOYL)-1H-BENZO[D]IMIDAZOL-2-YL)-PYRAZOL-5-CARBOXAMIDE] DERIVATIVES AND RELATED COMPOUNDS AS STING (STIMULATOR OF INTERFERON GENES) AGONISTS FOR THE TREATMENT OF CANCER Mersana Therapeutics, Inc. (US) 2022-06-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242531-A1 Monoacylglycerol Lipase Modulators MGLL, LPL, PNLIP KDM4E 2800/4885CSNK2A1 1260/4885CSNK2A2 1047/4885
US-11993601-B2 Monoacylglycerol lipase modulators MGLL, LPL, PNLIP KDM4E 2800/4885CSNK2A1 1260/4885CSNK2A2 1047/4885
US-11597728-B2 Monoacylglycerol lipase modulators MGLL, LPL, PNLIP KDM4E 2800/4885CSNK2A1 1260/4885CSNK2A2 1047/4885
US-20220315583-A1 Monoacylglycerol Lipase Modulators MGLL, LPL, PNLIP KDM4E 2800/4885CSNK2A1 1260/4885CSNK2A2 1047/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.