Propiram

Propiram

SCHEMBL29725982

CCC(=O)N(c1ccccn1)C(C)CN1CCCCC1.O=C(O)/C=C/C(=O)O

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRB1ADRB2ATP4AATP4BAXLCHRM2CHRM3DRD2FLT3HRH1HTR2AHTR2BHTR2CKCNH2KMT2AMAP2K1MAP2K2MEN1MLNRPLK4RENS1PR1SLC6A2SLC6A4atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Propiram. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 known ✓ O00255 2/20 0.48
KMT2A known ✓ Q03164 2/20 0.48
HTR1A P08908 1/20 0.48
ACHE P22303 1/20 0.46
OPRM1 P35372 9/20 0.46
SIGMAR1 Q99720 1/20 0.41
LMNA P02545 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Propiram SCHEMBL11079155 1.00 MEN1 (0.48) MEN1KMT2AHTR1AACHEOPRM1
Propiram SCHEMBL592478 1.00 MEN1 (0.48) MEN1KMT2AHTR1AACHEOPRM1
Propiram SCHEMBL38655379 0.94 MEN1 (0.52) MEN1KMT2AHTR1AACHEOPRM1
Propiram SCHEMBL26193 0.94 MEN1 (0.52) MEN1KMT2AHTR1AACHEOPRM1
Propiram SCHEMBL3093165 0.92 MEN1 (0.52) MEN1KMT2AHTR1AACHEOPRM1
SCHEMBL26930970 0.80 OPRM1 (0.43) MEN1KMT2AHTR1AOPRM1SIGMAR1
Phenampromide SCHEMBL907886 0.78 OPRM1 (0.47) MEN1KMT2AOPRM1SMN1; SMN2
Phenampromide SCHEMBL907884 0.78 OPRM1 (0.47) MEN1KMT2AOPRM1SMN1; SMN2
Phenampromide SCHEMBL11661873 0.77 ALDH1A1 (0.49) MEN1KMT2AOPRM1SMN1; SMN2
Phenampromide SCHEMBL11661877 0.77 ALDH1A1 (0.49) MEN1KMT2AOPRM1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250152319-A1 ORAL APPLIANCE FOR DELIVERY OF MEDICAMENTS AND/OR OTHER SUBSTANCES Emanate Biomedical, Inc. (US) 2025-05-15 US disclosed
US-12296085-B2 Method for extracorporeal treatment of preeclampsia and related disorders ImMutriX Therapeutics, Inc. (US) 2025-05-13 US disclosed
US-20250049928-A1 ANESTHETIC PRODRUGS AND DERIVATIVES THEREOF FOR PROLONGED SENSORY SELECTIVE NERVE BLOCKAGE THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ALABAMA 2025-02-13 US disclosed
US-20250032221-A1 ORTHODONTIC DEVICES FOR DELIVERY OF AN ACTIVE AGENT Smylio Inc. (US) 2025-01-30 US disclosed
US-12207984-B2 Oral appliance for delivery of medicaments and/or other substances Emanate Biomedical, Inc. (US) 2025-01-28 US disclosed
CN-118613231-A Orthodontic device for delivering active agents 斯米利奥公司 2024-09-06 CN disclosed
US-20240294909-A1 AGENTS, COMPOSITIONS, AND METHODS FOR THE TREATMENT OF HYPOXIA AND ISCHEMIA-RELATED DISORDERS MERAND PHARMACEUTICALS INC (US) 2024-09-05 US disclosed
US-20240247313-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2024-07-25 US disclosed
CN-117280030-A Agents, compositions and methods for treating hypoxia and ischemia related conditions 梅兰德制药公司 2023-12-22 CN disclosed
EP-3423102-B1 COMPOSITION FOR USE IN THE TREATMENT OF PREECLAMPSIA IMMUTRIX THERAPEUTICS INC (US) 2022-09-07 EP disclosed
WO-2022174113-A1 AGENTS, COMPOSITIONS, AND METHODS FOR THE TREATMENT OF HYPOXIA AND ISCHEMIA-RELATED DISORDERS MERAND PHARMACEUTICALS, INC. (US) 2022-08-18 WO disclosed
US-20220220561-A1 METHODS AND CLINICAL PROTOCOLS AND KITS PERTAINING TO MAKING AND USING THERAPEUTIC COMPOSITIONS FOR CELLULAR TREATMENT Advanced ReGen Medical Technologies, LLC 2022-07-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240247313-A1 SEROTONIN TRANSPORTER GENE AND TREATMENT OF OPIOID-RELATED DISORDERS SLC6A4, SLC6A3, SLC6A2 MEN1 4859/4885KMT2A 1923/4885HTR1A 16/4885
US-20250049928-A1 ANESTHETIC PRODRUGS AND DERIVATIVES THEREOF FOR PROLONGED SENSORY SELECTIVE NERVE BLOCKAGE TRPV1, OPRL1, TRPA1 MEN1 4804/4885KMT2A 3880/4885HTR1A 505/4885
US-12296085-B2 Method for extracorporeal treatment of preeclampsia and related disorders TEK, FLT4, PGF MEN1 1127/4885KMT2A 2469/4885HTR1A 4099/4885
US-20220220561-A1 METHODS AND CLINICAL PROTOCOLS AND KITS PERTAINING TO MAKING AND USING THERAPEUTIC COMPOSITIONS FOR CELLULAR TREATMENT CD47, HAVCR2, BST2 MEN1 2574/4885KMT2A 4472/4885HTR1A 4604/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.