SCHEMBL30478686

SCHEMBL30478686

CN(C)C=Nc1ccc(C2=CCN(NC(=O)OC(C)(C)C)CC2)cc1C#N

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 1/20 0.33
NAMPT P43490 2/20 0.33
HTR1D P28221 2/20 0.32
HTR1B P28222 2/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
QDPR P09417 2/20 0.31
EED O75530 1/20 0.31
RBBP4 Q09028 1/20 0.31
SUZ12 Q15022 1/20 0.31
EZH2 Q15910 1/20 0.31
KMT2A Q03164 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RET P07949 1/20 0.30
EGLN2 Q96KS0 1/20 0.30
GPR119 Q8TDV5 1/20 0.30
LIPE Q05469 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30478691 1.00 TBK1 (0.33) TBK1NAMPTHTR1DHTR1BNR1H2
SCHEMBL29025865 0.87 KMT2A (0.35) NAMPTHTR1DHTR1BQDPRKMT2A
SCHEMBL29025867 0.87 KMT2A (0.35) NAMPTHTR1DHTR1BQDPRKMT2A
SCHEMBL30478687 0.85 NAMPT (0.45) TBK1NAMPTNR1H2NR1H3EED
SCHEMBL29025848 0.81 QDPR (0.41) NAMPTQDPRKMT2ASMN1; SMN2ALDH1A1
SCHEMBL29025852 0.81 QDPR (0.41) NAMPTQDPRKMT2ASMN1; SMN2ALDH1A1
SCHEMBL7677344 0.71 NAMPT (0.39) NAMPTHTR1DHTR1BKMT2ALIPE
SCHEMBL29025844 0.71 RAB9A (0.35) SMN1; SMN2RETEGLN2
SCHEMBL1368952 0.69 NAMPT (0.36) NAMPTHTR1DHTR1BGPR119LIPE
SCHEMBL25353312 0.69 ALDH1A1 (0.45) NAMPTNR1H2NR1H3KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109422755-B Nitrogen-containing heterocyclic compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2023-07-04 CN disclosed