SCHEMBL30529271

SCHEMBL30529271

O=c1cnn(Cc2cc(F)c(F)cc2F)c(=O)[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.42
GRIA2 P42262 1/20 0.42
GRIA4 P48058 1/20 0.42
GRIK5 Q16478 1/20 0.42
BTK Q06187 2/20 0.34
PKM P14618 8/20 0.33
PKLR P30613 6/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP12 P39900 1/20 0.33
ROCK2 O75116 1/20 0.33
PDE3A Q14432 2/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
TRAP1 Q12931 1/20 0.32
TSHR P16473 2/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30174383 0.73 PKM (0.55) GRIA1GRIA2GRIA4GRIK5PKM
SCHEMBL11086435 0.71 MEN1 (0.60) GRIA1GRIA2GRIA4GRIK5PKM
SCHEMBL30995454 0.70 MMP1 (0.43) PKMMMP1MMP2MMP9MMP12
SCHEMBL30020048 0.69 HSD17B10 (0.54) GRIA1GRIA2GRIA4GRIK5PKM
SCHEMBL30753174 0.69 TRAP1 (0.40) MMP1MMP2MMP9MMP12THRB
SCHEMBL9540945 0.69 GRIA1 (0.56) GRIA1GRIA2GRIA4GRIK5PDE3A
SCHEMBL12294592 0.69 GRIA1 (0.51) GRIA1GRIA2GRIA4GRIK5PDE3A
SCHEMBL24781783 0.68 THRA (0.35) GRIA1GRIA2GRIA4GRIK5PKM
SCHEMBL30529262 0.68 P2RX7 (0.36) BTKPKMPKLRHSP90AA1HSP90AB1
SCHEMBL24780765 0.67 THRB (0.43) THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023165459-A1 COMPOUNDS AS SARS-COV-2 INHIBITORS FOCHON BIOSCIENCES , LTD. (CN) 2023-09-07 WO disclosed