SCHEMBL30697188

SCHEMBL30697188

Nc1cc(C(=O)O)nc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
HIF1A Q16665 1/20 0.41
P2RX7 Q99572 1/20 0.40
ALDH1A1 P00352 3/20 0.40
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
ASPH Q12797 1/20 0.39
HSD17B10 Q99714 3/20 0.38
KDM4E B2RXH2 2/20 0.38
IRAK4 Q9NWZ3 1/20 0.37
RBP4 P02753 1/20 0.36
CDK8 P49336 1/20 0.36
CDK19 Q9BWU1 1/20 0.36
HPGD P15428 1/20 0.36
SYK P43405 1/20 0.35
POLB P06746 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
IGFBP3 P17936 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27077029 1.00 ALOX15 (0.41) ALOX15TSHRHIF1AP2RX7ALDH1A1
SCHEMBL22695513 0.85 LMNA (0.42) P2RX7ALDH1A1HSP90AA1HSP90AB1HSD17B10
SCHEMBL29882592 0.84 HSP90AA1 (0.42) P2RX7ALDH1A1HSP90AA1HSP90AB1HSD17B10
SCHEMBL18839634 0.84 HSP90AA1 (0.42) P2RX7ALDH1A1HSP90AA1HSP90AB1HSD17B10
SCHEMBL4086004 0.82 ALOX15 (0.35) ALOX15TSHRHIF1AASPHIGFBP3
SCHEMBL22540919 0.81 P2RX7 (0.59) P2RX7ALDH1A1HSP90AA1HSP90AB1KDM4E
SCHEMBL2342015 0.80 NQO2 (0.46) P2RX7ALDH1A1HSP90AA1HSP90AB1KDM4E
SCHEMBL745813 0.80 TSHR (0.61) ALOX15TSHRHIF1AALDH1A1ASPH
SCHEMBL742374 0.80 TSHR (0.61) ALOX15TSHRHIF1AALDH1A1ASPH
SCHEMBL12097960 0.79 CES2 (0.45) ALOX15TSHRHIF1AP2RX7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117098764-A Tetrahydrothienopyridine derivatives as DDR inhibitors 奇斯药制品公司 2023-11-21 CN disclosed
CN-117062812-A Indoline derivatives as DDR inhibitors 奇斯药制品公司 2023-11-14 CN disclosed