SCHEMBL314763

SCHEMBL314763

COCCOc1[c]cccc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
CA2 P00918 1/20 0.35
MPO P05164 1/20 0.34
USP8 P40818 1/20 0.33
KDM1A O60341 4/20 0.32
PKM P14618 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
ADRB2 P07550 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7779040 0.94 L3MBTL1 (0.37) TSHRCA2MPOSMN1; SMN2
SCHEMBL6132567 0.90 KCNA3 (0.35) TSHRSMN1; SMN2
SCHEMBL1143957 0.90 SMN1; SMN2 (0.38) TSHRSMN1; SMN2
SCHEMBL6238419 0.89 JAK2 (0.33) SMN1; SMN2
SCHEMBL6132896 0.89 KDM4E (0.35) SMN1; SMN2
SCHEMBL4813845 0.85 TSHR (0.33) TSHRCA2MPO
SCHEMBL2453704 0.82 DRD2 (0.46) TSHRSMN1; SMN2
SCHEMBL757705 0.82 PTPN1 (0.37) SMN1; SMN2
SCHEMBL126227 0.82 ALDH1A1 (0.34) CA2SMN1; SMN2
SCHEMBL2449865 0.81 L3MBTL1 (0.38) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 777 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4330247-A1 COMPOUNDS AND THEIR USES AS CD38 INHIBITORS Nanjing Immunophage Biotech Co., Ltd (CN) 2024-03-06 EP claimed
WO-2022228496-A1 COMPOUNDS AND THEIR USES AS CD38 INHIBITORS NANJING IMMUNOPHAGE BIOTECH CO., LTD (CN) 2022-11-03 WO claimed
WO-2021078120-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES NOVARTIS AG (CH) 2021-04-29 WO claimed
EP-2951179-B1 SPIRO-QUINAZOLINONE DERIVATIVES USEFUL FOR THE TREATMENT OF NEUROLOGICAL DISEASES AND CONDITIONS MERCK PATENT GMBH (DE) 2020-03-11 EP claimed
US-9708321-B2 Spiro-quinazolinone derivatives and their use as positive allosteric modulators of mGluR4 MERCK PATENT GMBH (DE) 2017-07-18 US claimed
CN-105121455-B Novel triptolide derivative and preparation method and application thereof 香港浸会大学 2017-06-16 CN claimed
US-20150361079-A1 Spiro-Quinazolinone Derivatives and their Use as Positive Allosteric Modulators of mGluR4 MERCK PATENT GMBH (DE) 2015-12-17 US claimed
EP-2951179-A1 SPIRO-QUINAZOLINONE DERIVATIVES USEFUL FOR THE TREATMENT OF NEUROLOGICAL DISEASES AND CONDITIONS Merck Patent GmbH (DE) 2015-12-09 EP claimed
CN-102781937-B As two (difluoromethyl) pyrazoles of sterilant BAYER CROPSCIENCE AG (DE) 2015-09-30 CN claimed
EP-2516426-B1 BIS(DIFLUORMETHYL)PYRAZOLES USED AS FUNGICIDES BAYER CROPSCIENCE AG (DE) 2015-09-16 EP claimed
WO-2010139731-A1 1H-IMIDAZO[4,5-c]QUINOLINONE DERIVATIVES NOVARTIS AG (CH) 2010-12-09 WO claimed
EP-1036062-B1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE (MMP) INHIBITORS PFIZER LTD (GB) 2004-01-02 EP claimed
US-6495568-B1 TREATMENT OF TISSUE ULCERATION, WOUND REPAIR AND SKIN DISEASES WARNER-LAMBERT COMPANY 2002-12-17 US claimed
CN-1281433-A Hydroxamic acid derivatives as matrix metalloproteinase (MMP) inhibitors PFIZER LTD (US) 2001-01-24 CN claimed
EP-1036062-A1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE (MMP) INHIBITORS Pfizer Limited (GB) 2000-09-20 EP claimed
WO-1999029667-A1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE (MMP) INHIBITORS PFIZER LIMITED (GB) 1999-06-17 WO claimed
EP-0367887-B1 Herbicidal concentrate CIBA GEIGY AG (CH) 1994-03-30 EP claimed
US-4933000-A Herbicidal compound concentrate CIBA-GEIGY CORPORATION (US) 1990-06-12 US claimed
EP-0367887-A2 Herbicidal concentrate CIBA-GEIGY AG (CH) 1990-05-16 EP claimed
EP-0348343-A2 Synergistic agent and process for selective weed control in cereals, maize and rice CIBA-GEIGY AG (CH) 1989-12-27 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150361079-A1 Spiro-Quinazolinone Derivatives and their Use as Positive Allosteric Modulators of mGluR4 GRM4, GRIA4, GRIK4 TSHR 839/4885CA2 2342/4885MPO 4818/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.