SCHEMBL315077

SCHEMBL315077

CN(C)C1(Cc2ccccc2)CCC(NC(=O)c2noc3c2CN(S(=O)(=O)Cc2cccc(C(F)(F)F)c2)CC3)CC1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.38
TRPV1 Q8NER1 3/20 0.38
SIGMAR1 Q99720 2/20 0.37
SMYD3 Q9H7B4 1/20 0.37
GPR52 Q9Y2T5 2/20 0.37
UBE2M P61081 3/20 0.36
DCUN1D1 Q96GG9 3/20 0.36
DRD4 P21917 2/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
GPR142 Q7Z601 1/20 0.36
KMT2A Q03164 1/20 0.35
HSP90AA1 P07900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5246034 0.80 GPR142 (0.46) UBE2MDCUN1D1MAPTTHRBGPR142
SCHEMBL325035 0.80 ALDH1A1 (0.40) MAPTKMT2A
SCHEMBL5246039 0.73 GPR142 (0.44) UBE2MDCUN1D1MAPTTHRBGPR142
SCHEMBL2582295 0.69 GAA (0.42) KMT2A
SCHEMBL2581672 0.68 DRD4 (0.53) SIGMAR1DRD4
SCHEMBL4261853 0.66 LMNA (0.48) MAPTTHRB
SCHEMBL2582296 0.65 CRHBP (0.44) OPRM1MAPTTHRBKMT2A
SCHEMBL1944694 0.64 DRD4 (0.44) SIGMAR1SMYD3GPR52UBE2MDCUN1D1
SCHEMBL2585658 0.63 CCR2 (0.46) SMYD3DRD4
SCHEMBL315901 0.63 ALDH1A1 (0.52) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed
US-20070129369-A1 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070129369-A1 Heteroaryl substituted cyclohexyl-1,4-diamine compounds DDC, DPYD, PKD1 OPRM1 2315/4885TRPV1 4251/4885SIGMAR1 2685/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.