SCHEMBL315514

SCHEMBL315514

OB(O)c1cncc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.43
ENPP2 Q13822 1/20 0.42
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
TTR P02766 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2557007 0.82 GAA (0.42) CHRNB2CHRNA4
SCHEMBL28967087 0.82 ENPP2 (0.36) ENPP2TTR
SCHEMBL13651757 0.73 ENPP2 (0.44) ENPP2TTRCHRNB2CHRNA4
SCHEMBL29538949 0.73 HCAR2 (0.45) HCAR2ENPP2
SCHEMBL29957005 0.73 ENPP2 (0.44) ENPP2TTRCHRNB2CHRNA4
SCHEMBL27969 0.73 HCAR2 (0.45) HCAR2ENPP2
SCHEMBL25098761 0.73 CHRNB2 (0.35) HCAR2CHRNB2CHRNA4
SCHEMBL197638 0.73
Hydrochloric Acid SCHEMBL16899234 0.71 ENPP2 (0.43) ENPP2TTRCHRNB2CHRNA4
SCHEMBL144194 0.71 HCAR2 (0.43) HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 699 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111116559-A Pyridine urea compound and preparation method and pharmaceutical application thereof 复旦大学 2020-05-08 CN claimed
US-9156834-B2 Derivatives of heteroarylsulfonamides, their preparation and their application in human therapy PIERRE FABRE MEDICAMENT (FR) 2015-10-13 US claimed
US-20140357624-A1 DERIVATIVES OF HETEROARYLSULFONAMIDES, THEIR PREPARATION AND THEIR APPLICATION IN HUMAN THERAPY PF MEDICAMENT (FR) 2014-12-04 US claimed
US-8846930-B2 Derivatives of heteroarylsulfonamides, their preparation and their application in human therapy PIERRE FABRE MEDICAMENT (FR) 2014-09-30 US claimed
EP-2643318-A1 DERIVATIVES OF HETEROARYLSULFONAMIDES, THEIR PREPARATION AND THEIR APPLICATION IN HUMAN THERAPY Pierre Fabre Médicament (FR) 2013-10-02 EP claimed
US-20130172326-A1 DERIVATIVES OF HETEROARYLSULFONAMIDES, THEIR PREPARATION AND THEIR APPLICATION IN HUMAN THERAPY PIERRE FABRE MEDICAMENT (FR) 2013-07-04 US claimed
WO-2012069503-A1 DERIVATIVES OF HETEROARYLSULFONAMIDES, THEIR PREPARATION AND THEIR APPLICATION IN HUMAN THERAPY PIERRE FABRE MEDICAMENT (FR) 2012-05-31 WO claimed
US-20260125392-A1 URACIL DERIVATIVES HAVING VIRUS REPLICATION INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME SHIONOGI & CO., LTD. (JP) 2026-05-07 US disclosed
US-12617802-B2 Sulfonimidamide compounds as NLRP3 modulators GENENTECH, INC. (US) 2026-05-05 US disclosed
EP-4568746-B1 BICYCLIC TETRAHYDROTHIAZEPINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2026-04-29 EP disclosed
US-20260098036-A1 2-HETEROARYL-3-OXO-2,3-DIHYDROPYRIDAZINE-4-CARBOXAMIDES FOR THE TREATMENT OF CANCER DEUTSCHES KREBSFORSCHUNGSZENTRUM (DE) 2026-04-09 US disclosed
US-20260070932-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF ANNEXON INC (US) 2026-03-12 US disclosed
US-12545687-B2 Uracil derivatives having virus replication inhibitory activity and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2026-02-10 US disclosed
US-20090182013-A1 Derivatives of 5-Thioxylopyranose and Use of Same for Treatment LABORATOIRES FOURNIER S.A. (FR) 2009-07-16 US disclosed
WO-2009074246-A1 NOVEL 2-HETARYL THIAZOLE-4-CARBOXAMIDE DERIVATIVES, PRODUCTION THEREOF, AND USE THEREOF AS A MEDICAMENT BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-06-18 WO disclosed
EP-2070924-A1 New 2 hetarylthiazol-4-carboxylic acid derivatives, their manufacture and use as medicine Bayer Schering Pharma Aktiengesellschaft (DE) 2009-06-17 EP disclosed
WO-2009017664-A1 CYCLIC INHIBITORS OF 11β-HYDROXYSTERIOD DEHYDROGENASE 1 VITAE PHARMACEUTICALS, INC. (US) 2009-02-05 WO disclosed
US-20080176862-A1 Cognitive impairment, Alzheimer disease, neurodegeneration, dementia; such as 3'-(2-amino-4-(2-chloropyridin-4-yl)-1-methyl-5-oxo-4,5-dihydro-1H-imidazol-4-yl)-5-chlorobiphenyl-3-yl methanesulfonate; Beta site APP Cleaving Enzyme (BACE) inhibitors ASTRAZENECA AB (SE) 2008-07-24 US disclosed
US-20080161269-A1 Compounds 620 ASTRAZENECA AB (SE) 2008-07-03 US disclosed
US-5629428-A 3-Chloropyridines, and their use in liquid-crystal mixtures HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161269-A1 Compounds 620 MAPT, PSEN1, PSEN2 HCAR2 1487/4885ENPP2 3174/4885MKNK1 437/4885
US-20080176862-A1 Cognitive impairment, Alzheimer disease, neurodegeneration, dementia; such as 3'-(2-amino-4-(2-chloropyridin-4-yl)-1-methyl-5-oxo-4,5-dihydro-1H-imidazol-4-yl)-5-chlorobiphenyl-3-yl methanesulfonate; Beta site APP Cleaving Enzyme (BACE) inhibitors BACE1, BACE2, PSEN1 HCAR2 3311/4885ENPP2 3267/4885MKNK1 763/4885
US-20260125392-A1 URACIL DERIVATIVES HAVING VIRUS REPLICATION INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME SARS1, ACE, RNGTT HCAR2 4567/4885ENPP2 4801/4885MKNK1 3775/4885
US-20260098036-A1 2-HETEROARYL-3-OXO-2,3-DIHYDROPYRIDAZINE-4-CARBOXAMIDES FOR THE TREATMENT OF CANCER AHR, CBR1, CNR1 HCAR2 10/4885ENPP2 2252/4885MKNK1 3789/4885
US-20130172326-A1 DERIVATIVES OF HETEROARYLSULFONAMIDES, THEIR PREPARATION AND THEIR APPLICATION IN HUMAN THERAPY KCNA4, KCNA1, KCNB1 HCAR2 653/4885ENPP2 3252/4885MKNK1 1732/4885
US-12617802-B2 Sulfonimidamide compounds as NLRP3 modulators NLRP3, NLRP1, PYCARD HCAR2 463/4885ENPP2 4253/4885MKNK1 2425/4885
US-20140357624-A1 DERIVATIVES OF HETEROARYLSULFONAMIDES, THEIR PREPARATION AND THEIR APPLICATION IN HUMAN THERAPY KCNA4, KCNA1, KCNB1 HCAR2 653/4885ENPP2 3252/4885MKNK1 1732/4885
US-20260070932-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF CFH, CFB, C5 HCAR2 374/4885ENPP2 34/4885MKNK1 3311/4885
US-20090182013-A1 Derivatives of 5-Thioxylopyranose and Use of Same for Treatment TPMT, PNPO, PPOX HCAR2 3232/4885ENPP2 545/4885MKNK1 3785/4885
US-12545687-B2 Uracil derivatives having virus replication inhibitory activity and pharmaceutical composition comprising the same SARS1, ACE, ACE2 HCAR2 3842/4885ENPP2 4653/4885MKNK1 3011/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.