SCHEMBL3246424

SCHEMBL3246424

NC(=O)c1cccc(COC(=O)N(CCN2CCC(c3cn[nH]c3)C2)c2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.43
HSD11B1 P28845 3/20 0.41
OPRK1 P41145 2/20 0.38
PTGIR P43119 1/20 0.38
OPRM1 P35372 5/20 0.38
SIGMAR1 Q99720 1/20 0.38
CHRM5 P08912 2/20 0.37
CHRM1 P11229 2/20 0.37
CHRM3 P20309 2/20 0.37
ACHE P22303 1/20 0.37
CHRM2 P08172 1/20 0.37
OPRD1 P41143 2/20 0.36
PARP1 P09874 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3246422 0.79 ROCK2 (0.49)
SCHEMBL4465185 0.64 MEN1 (0.55) CCR5SIGMAR1ACHEKMT2A
SCHEMBL31572354 0.61 ALDH1A1 (0.52) HSD11B1ALDH1A1
Hydrochloric Acid SCHEMBL19580057 0.60 HTR7 (0.52) OPRM1SIGMAR1OPRD1KMT2A
SCHEMBL27150592 0.59 HSD11B1 (0.57) HSD11B1ALDH1A1
SCHEMBL27150593 0.59 HSD11B1 (0.57) HSD11B1ALDH1A1
SCHEMBL3245955 0.59 ROCK2 (0.48)
SCHEMBL12311314 0.59 PAX8 (0.49) CHRM5CHRM1CHRM3CHRM2ALDH1A1
SCHEMBL433443 0.58 HRH3 (0.43) OPRK1PTGIROPRM1SIGMAR1OPRD1
SCHEMBL25920399 0.58 CHRM2 (0.43) CHRM1CHRM3CHRM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed