SCHEMBL329312

SCHEMBL329312

Clc1ccc2c(c1)CNC2

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 4/20 0.69
HTR2C P28335 7/20 0.56
HTR2A P28223 6/20 0.56
HTR2B P41595 5/20 0.56
ASIC3 Q9UHC3 1/20 0.44
AHR P35869 2/20 0.41
CMA1 P23946 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
SLC6A4 P31645 2/20 0.40
ADRB1 P08588 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CNR1 P21554 1/20 0.40
SLC6A2 P23975 1/20 0.40
HRH1 P35367 1/20 0.40
KCNH2 Q12809 1/20 0.40
METAP1 P53582 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL383414 0.98 PNMT (0.67) PNMTHTR2CHTR2AHTR2BASIC3
Bromide SCHEMBL949591 0.98 PNMT (0.67) PNMTHTR2CHTR2AHTR2BASIC3
Hydrochloric Acid SCHEMBL16033643 0.95 PNMT (0.64) PNMTHTR2CHTR2AHTR2BASIC3
SCHEMBL532012 0.82 PNMT (0.85) PNMTHTR2CHTR2AHTR2BASIC3
SCHEMBL329775 0.82 PNMT (1.00) PNMTHTR2CHTR2AHTR2BASIC3
SCHEMBL29543416 0.82 ASIC3 (0.56) PNMTHTR2CHTR2AHTR2BASIC3
SCHEMBL29587836 0.82 PNMT (1.00) PNMTHTR2CHTR2AHTR2BASIC3
Hydrochloric Acid SCHEMBL947776 0.81 PNMT (0.81) PNMTHTR2CHTR2AHTR2BASIC3
Hydrochloric Acid SCHEMBL1124954 0.81 PNMT (0.96) PNMTHTR2CHTR2AHTR2BASIC3
SCHEMBL25207974 0.79 PNMT (0.79) PNMTHTR2CHTR2AHTR2BASIC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 252 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4731626-A1 PI3K INHIBITORS AND USE THEREOF Regor Pharmaceuticals, Inc. (US) 2026-04-29 EP disclosed
EP-3704125-B1 MODULATORS OF THE INTEGRATED STRESS PATHWAY CALICO LIFE SCIENCES LLC (US) 2026-03-11 EP disclosed
US-20260034127-A1 TREATMENT OF GVHD KADMON CORP LLC (FR) 2026-02-05 US disclosed
US-20250144094-A1 THIOPHENE ULK1/2 INHIBITORS AND THEIR USE THEREOF ERASCA, INC. 2025-05-08 US disclosed
WO-2024260464-A1 PI3K INHIBITORS AND USE THEREOF REGOR PHARMACEUTICALS, INC. (US) 2024-12-26 WO disclosed
EP-4433059-A1 THIOPHENE ULK1/2 INHIBITORS AND THEIR USE THEREOF Erasca, Inc. (US) 2024-09-25 EP disclosed
CN-114072398-B Compounds that inhibit TDG activity 上海仕谱生物科技有限公司 2024-06-11 CN disclosed
US-20240174631-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR MODULATING FGF ACTIVITY RECOVERY THERAPEUTICS, INC. 2024-05-30 US disclosed
US-11939320-B2 Modulators of the integrated stress pathway ABBVIE INC. (US) 2024-03-26 US disclosed
EP-4291177-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR MODULATING FGF ACTIVITY Recovery Therapeutics, Inc. (US) 2023-12-20 EP disclosed
CN-1162424-C Quinoline-4-radical derivative II - 2004-08-18 CN disclosed
EP-1343796-A2 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2003-09-17 EP disclosed
WO-2002034760-A2 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2002-05-02 WO disclosed
US-6339093-B1 Isoquinoline derivatives HOFFMANN-LA ROCHE INC. 2002-01-15 US disclosed
CN-1304936-A Quinoline-4-radical derivative II HOFFMANN LA BOCHE & CO AG F (CH) 2001-07-25 CN disclosed
EP-1090917-A1 Quinolin-4-yl derivatives and their use as NMDA-receptor subtype blockers F. HOFFMANN-LA ROCHE AG (CH) 2001-04-11 EP disclosed
US-5726197-A ADRENORECEPTORS AND ADMINISTERING SYNTEX (U.S.A.) INC. (US) 1998-03-10 US disclosed
US-5026856-A Bactericides WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1991-06-25 US disclosed
EP-0343560-A2 Isoindoline derivative WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1989-11-29 EP disclosed
EP-0056144-A1 Carboxylic acid derivatives, their preparation and use as pharmaceuticals Dr. Karl Thomae GmbH (DE) 1982-07-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250144094-A1 THIOPHENE ULK1/2 INHIBITORS AND THEIR USE THEREOF ULK1, ULK2, ULK3 PNMT 2917/4885HTR2C 2564/4885HTR2A 2807/4885
US-20260034127-A1 TREATMENT OF GVHD ROCK2, RHOA, MYH2 PNMT 2804/4885HTR2C 4007/4885HTR2A 4112/4885
US-20240174631-A1 COMPOUNDS, COMPOSITIONS, AND METHODS FOR MODULATING FGF ACTIVITY FGF1, FGF2, FGFR1 PNMT 4852/4885HTR2C 1517/4885HTR2A 1239/4885
US-11939320-B2 Modulators of the integrated stress pathway ATF4, ATF1, DDIT3 PNMT 1437/4885HTR2C 1925/4885HTR2A 1445/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.