SCHEMBL3341844

SCHEMBL3341844

COc1ccc(CC(C)NCc2ccccc2)cc1.CS(=O)(=O)O

nearest known ligand 0.66

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.62
HTT P42858 1/20 0.57
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.55
ALDH1A1 P00352 4/20 0.51
NPC1 O15118 1/20 0.50
MMP1 P03956 1/20 0.49
MMP9 P14780 1/20 0.49
MMP13 P45452 1/20 0.49
SLC2A1 P11166 1/20 0.48
MAPK1 P28482 1/20 0.48
POLB P06746 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3341840 1.00 SIGMAR1 (0.62) SIGMAR1HTTMEN1KMT2AL3MBTL1
SCHEMBL3346880 1.00 SIGMAR1 (0.62) SIGMAR1HTTMEN1KMT2AL3MBTL1
SCHEMBL593666 0.92 SIGMAR1 (0.74) SIGMAR1HTTMEN1KMT2AL3MBTL1
SCHEMBL8092326 0.92 SIGMAR1 (0.74) SIGMAR1HTTMEN1KMT2AL3MBTL1
SCHEMBL2795948 0.92 SIGMAR1 (0.74) SIGMAR1HTTMEN1KMT2AL3MBTL1
SCHEMBL719011 0.92 SIGMAR1 (0.74) SIGMAR1HTTMEN1KMT2AL3MBTL1
Hydrochloric Acid SCHEMBL1134233 0.90 SIGMAR1 (0.72) SIGMAR1HTTMEN1KMT2AL3MBTL1
Hydrochloric Acid SCHEMBL1134234 0.90 SIGMAR1 (0.72) SIGMAR1HTTMEN1KMT2AL3MBTL1
SCHEMBL6539539 0.90 SIGMAR1 (0.59) SIGMAR1HTTMEN1KMT2AL3MBTL1
SCHEMBL3630860 0.86 SIGMAR1 (0.57) SIGMAR1MEN1KMT2AL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2172443-B1 METHOD FOR PRODUCING OPTICALLY ACTIVE AMINE HAMARI CHEMICALS LTD (JP) 2013-03-27 EP disclosed
US-8222452-B2 Method for producing optically active amines HAMARI CHEMICALS, LTD. (JP) 2012-07-17 US disclosed
US-20100160636-A1 METHOD FOR PRODUCING OPTICALLY ACTIVE AMINES HAMARI CHEMICALS, LTD. (JP) 2010-06-24 US disclosed
EP-2172443-A1 METHOD FOR PRODUCING OPTICALLY ACTIVE AMINE Hamari Chemicals, Ltd. (JP) 2010-04-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100160636-A1 METHOD FOR PRODUCING OPTICALLY ACTIVE AMINES INMT, HNMT, PADI3 SIGMAR1 943/4885HTT 527/4885MEN1 1082/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.