SCHEMBL3351014

SCHEMBL3351014

O=C(O)c1cccc2c1OC(F)(F)C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.40
PKM P14618 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ALDH1A1 P00352 5/20 0.40
MAPT P10636 1/20 0.40
KDM4E B2RXH2 3/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 2/20 0.37
ALB P02768 1/20 0.37
PARP1 P09874 1/20 0.36
NR4A1 P22736 1/20 0.34
NR4A2 P43354 1/20 0.34
NR4A3 Q92570 1/20 0.34
CXCR5 P32302 1/20 0.34
HSD17B10 Q99714 2/20 0.33
HPGD P15428 2/20 0.33
CYP2D6 P10635 1/20 0.33
G6PD P11413 1/20 0.33
CASP7 P55210 1/20 0.33
CASP6 P55212 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL783714 0.80 LMNA (0.59) LMNAPKMNPSR1ALDH1A1MAPT
SCHEMBL7413765 0.78 FFAR4 (0.42) LMNAPKMNPSR1ALDH1A1MAPT
SCHEMBL2548565 0.78 LMNA (0.44) LMNAPKMNPSR1ALDH1A1MAPT
SCHEMBL15625037 0.71 PKM (0.39) LMNAPKMNPSR1ALDH1A1MAPT
SCHEMBL672668 0.71 LMNA (0.44) LMNAPKMNPSR1ALDH1A1MAPT
SCHEMBL21845449 0.70 TRPA1 (0.42) ALDH1A1ALOX15TSHRALBCXCR5
SCHEMBL11094419 0.69 PARP1 (0.49) ALDH1A1MAPTKDM4EALOX15TSHR
SCHEMBL11797726 0.69 ALDH1A1 (0.44) ALDH1A1KDM4EALOX15TSHRALB
SCHEMBL29710998 0.69 ALOX5 (0.41) ALDH1A1KDM4EALOX15TSHRALB
SCHEMBL14297655 0.69 GABRA1 (0.36) LMNATSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038200-A1 OXAZOLIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2010-04-08 WO claimed
WO-2010038200-A1 OXAZOLIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2010-04-08 WO disclosed