SCHEMBL3358868

SCHEMBL3358868

CN1CCN(Cc2cn(C)c3cc(N)ccc23)CC1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.53
LMNA P02545 2/20 0.50
GLA P06280 1/20 0.49
HTR6 P50406 14/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
HRH3 Q9Y5N1 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3352639 0.89 NR1H2 (0.53) NR1H2LMNAGLAHTR6ALDH1A1
SCHEMBL3353653 0.89 ACHE (0.50) NR1H2LMNAGLAALDH1A1TSHR
SCHEMBL3358110 0.86 HRH3 (0.55) NR1H2LMNAGLAALDH1A1TSHR
SCHEMBL3357970 0.82 NR1H2 (0.47) NR1H2LMNAHTR6ALDH1A1
SCHEMBL3354038 0.81 NR1H2 (0.46) NR1H2LMNAHTR6CYP3A4CYP2D6
SCHEMBL13537525 0.80 LMNA (0.46) LMNAGLAHTR6ALDH1A1TSHR
SCHEMBL3353571 0.78 ACHE (0.51) NR1H2LMNAGLAALDH1A1TSHR
SCHEMBL3356418 0.78 HTR6 (0.54) LMNAGLAHTR6
SCHEMBL2075509 0.77 HTR2A (0.44) HTR6HRH3
SCHEMBL3350921 0.77 ACHE (0.50) NR1H2LMNAGLAALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2141163-A1 Substituted thiazolidinones, their production and utilisation as medicine Bayer Schering Pharma AG (DE) 2010-01-06 EP disclosed
EP-2141163-A1 Substituted thiazolidinones, their production and utilisation as medicine Bayer Schering Pharma AG (DE) 2010-01-06 EP disclosed