SCHEMBL3467249

SCHEMBL3467249

N#Cc1cccc(-c2ccc(CCC(CCCc3ccc(OCc4ccccc4)cc3)C(=O)O)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 2/20 0.54
MMP13 P45452 2/20 0.54
FFAR1 O14842 7/20 0.53
FFAR4 Q5NUL3 2/20 0.53
AKR1B1 P15121 2/20 0.53
GPR34 Q9UPC5 4/20 0.52
PTGER4 P35408 1/20 0.48
PTGER3 P43115 1/20 0.48
ADAMTS4 O75173 1/20 0.47
FOLH1 Q04609 1/20 0.46
MMP2 P08253 1/20 0.45
MMP3 P08254 1/20 0.45
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
MAOB P27338 1/20 0.44
NR4A2 P43354 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7932591 0.92 MMP12 (0.63) MMP12MMP13FFAR1ADAMTS4FOLH1
SCHEMBL3466325 0.91 FFAR1 (0.57) MMP12MMP13FFAR1FFAR4AKR1B1
SCHEMBL7928277 0.91 MMP12 (0.64) MMP12MMP13FFAR1ADAMTS4FOLH1
SCHEMBL3467000 0.91 MMP12 (0.51) MMP12MMP13FFAR1FFAR4AKR1B1
SCHEMBL7928937 0.88 MMP12 (0.54) MMP12MMP13FFAR1FFAR4FOLH1
SCHEMBL1856449 0.84 LTA4H (0.60) MMP12FFAR1FFAR4MMP2MMP3
SCHEMBL3466565 0.84 GPR34 (0.54) MMP12MMP13FFAR1FFAR4AKR1B1
SCHEMBL3467017 0.83 MMP12 (0.57) MMP12MMP13FFAR1FFAR4ADAMTS4
SCHEMBL1858749 0.83 FOLH1 (0.50) MMP12MMP13FFAR1FFAR4GPR34
SCHEMBL7922593 0.82 MMP12 (0.56) MMP12MMP13FOLH1MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010070076-A1 ALKANOIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE AS HDAC INHIBITORS CRYSTAX PHARMACEUTICALS, S.L. (ES) 2010-06-24 WO claimed
WO-2010070076-A1 ALKANOIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE AS HDAC INHIBITORS CRYSTAX PHARMACEUTICALS, S.L. (ES) 2010-06-24 WO disclosed