SCHEMBL3530635

SCHEMBL3530635

N#CCC1(c2cccc(Cl)c2F)CCN(C(=O)O)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.39
JAK2 O60674 2/20 0.35
JAK1 P23458 2/20 0.35
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
DRD2 P14416 2/20 0.33
CYP3A4 P08684 2/20 0.32
USP2 O75604 1/20 0.32
CYP2D6 P10635 1/20 0.32
ALDH1A1 P00352 2/20 0.32
ALOX15 P16050 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32
EPHX2 P34913 1/20 0.32
CYP1A2 P05177 1/20 0.32
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5371500 0.78 DRD2 (0.44) DRD2ALDH1A1EPHX2
SCHEMBL3530123 0.78 APP (0.43) KDM1AJAK2JAK1CYP2C19P2RX7
SCHEMBL3530638 0.76 SLC6A4 (0.43) JAK2JAK1MAPT
SCHEMBL3528335 0.76 SLC6A3 (0.43) JAK2JAK1CYP3A4CYP2C19
SCHEMBL1245009 0.76 CRHBP (0.39) KMT2ADRD2CYP2D6ALDH1A1EPHX2
SCHEMBL2530864 0.74 DRD2 (0.40) KMT2ADRD2ALDH1A1EPHX2
SCHEMBL1243013 0.73 RIPK1 (0.38) MAPTKMT2AALOX15KDM4E
SCHEMBL6153201 0.72 METAP2 (0.38) DRD2CYP3A4USP2CYP2D6ALDH1A1
SCHEMBL2530292 0.70 SOS1 (0.36) DRD2CYP3A4USP2ALDH1A1ALOX15
SCHEMBL3526611 0.68 ALDH1A1 (0.48) KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed
US-20060229336-A1 Ccr5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORPORATION 2006-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060229336-A1 Ccr5 antagonists as therapeutic agents CCR5, CCR1, CXCR3 KDM1A 4598/4885JAK2 2862/4885JAK1 2938/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.