SCHEMBL3547636

SCHEMBL3547636

O=c1c(NCCCCc2ccccc2)c(-c2ccccc2)sn1CCc1cccc(F)c1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.39
ASAH1 Q13510 2/20 0.38
CACNA1G O43497 1/20 0.38
CACNA1H O95180 1/20 0.38
MAPT P10636 2/20 0.37
TP53 P04637 1/20 0.37
PRKCA P17252 1/20 0.36
GSK3B P49841 1/20 0.36
CASP7 P55210 1/20 0.36
FAAH O00519 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5184329 0.81 TYMP (0.42) CASP3ASAH1FAAH
SCHEMBL17844195 0.74 ASPH (0.41) ASAH1
SCHEMBL5184337 0.73 MAOA (0.42) ASAH1
SCHEMBL17844110 0.73 MAOA (0.40) ASAH1
SCHEMBL2001616 0.71 CA12 (0.40) ASAH1CACNA1GCACNA1HMAPT
SCHEMBL17844245 0.71 CYP1A2 (0.42) CASP7
SCHEMBL17844216 0.70 EPHX1 (0.40) ASAH1GSK3B
SCHEMBL5186011 0.68 ALDH1A1 (0.48) MAPTTP53FAAH
SCHEMBL17844169 0.66 SCN9A (0.36)
SCHEMBL17844161 0.66 FAAH (0.44) MAPTTP53CASP7FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7723333-B2 Non-anilinic derivatives of isothiazol-3(2H)-one 1,1-dioxides as liver X receptor modulators ASTRAZENECA AB (SE) 2010-05-25 US claimed
WO-2016100619-A2 TREATMENT AND DIAGNOSIS OF CANCER RGENIX, INC. (US) 2016-06-23 WO disclosed