SCHEMBL355358

SCHEMBL355358

Cc1ncccc1C(O)=S

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.52
KDM4E B2RXH2 3/20 0.42
TDP1 Q9NUW8 1/20 0.42
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
MAPT P10636 2/20 0.41
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
BLM P54132 1/20 0.41
AGER Q15109 1/20 0.41
MYC P01106 1/20 0.41
NAPRT Q6XQN6 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 2/20 0.39
GAA P10253 2/20 0.37
MKNK1 Q9BUB5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1375608 0.98 P2RX7 (0.50) P2RX7KDM4ETDP1NPC1RAB9A
SCHEMBL5740191 0.83 P2RX7 (0.52) P2RX7KDM4ETDP1NPC1RAB9A
SCHEMBL22734836 0.81 P2RX7 (0.55) P2RX7KDM4ETDP1NPC1RAB9A
SCHEMBL5073329 0.81 P2RX7 (0.55) P2RX7KDM4ETDP1NPC1RAB9A
SCHEMBL17210751 0.78 P2RX7 (0.52) P2RX7KDM4ETDP1NPC1RAB9A
SCHEMBL71547 0.78 KDM4E (0.63) P2RX7KDM4ETDP1NPC1RAB9A
SCHEMBL29651292 0.78 KDM4E (0.63) P2RX7KDM4ETDP1NPC1RAB9A
SCHEMBL30599010 0.78 P2RX7 (0.51) P2RX7KDM4ETDP1NPC1RAB9A
SCHEMBL29086505 0.78 P2RX7 (0.51) P2RX7KDM4ETDP1NPC1RAB9A
Acetic Acid SCHEMBL27987140 0.77 P2RX7 (0.56) P2RX7KDM4ETDP1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119707919-A Deuterated piperazine compound and preparation method and application thereof 山东大学 2025-03-28 CN claimed
WO-2006091506-A2 NEUROPEPTIDE Y4 RECEPTOR AGONISTS BAYER PHARMACEUTICALS CORPORATION (US) 2006-08-31 WO claimed
CN-119707919-A Deuterated piperazine compound and preparation method and application thereof 山东大学 2025-03-28 CN disclosed
CN-116874418-A Process for preparing 2- (methylsulfonyl) nicotinaldehyde 苏州源起材料科技有限公司 2023-10-13 CN disclosed
US-20230108636-A1 COMPOSITIONS AND METHODS FOR ENHANCING TRANSPORT THROUGH MUCUS UNIV JOHNS HOPKINS (US) 2023-04-06 US disclosed
EP-2200440-B1 ANTIBACTERIAL AMIDE AND SULFONAMIDE SUBSTITUTED HETEROCYCLIC UREA COMPOUNDS CRESTONE INC (US) 2017-07-19 EP disclosed
US-8148380-B2 Antibacterial amide and sulfonamide substituted heterocyclic urea compounds CRESTONE, INC. (US) 2012-04-03 US disclosed
US-20120015941-A1 Antibacterial Amide and Sulfonamide Substituted Heterocyclic Urea Compounds CRESTONE, INC. (US) 2012-01-19 US disclosed
US-20090280106-A1 Pituitary adenylate cyclase acivating peptide (pacap) receptor (vpac2) agonists and their pharmacological methods of use BAYER PHARMACEUTICALS CORPORATION (US) 2009-11-12 US disclosed
EP-1689421-A4 SELECTIVE NEUROPEPTIDE Y2 RECEPTOR AGONISTS BAYER HEALTHCARE AG (DE) 2009-06-24 EP disclosed
US-20090105122-A1 Selective neuropeptide y2 receptor agonists BAYER PHARMACEUTICALS CORPORATION (US) 2009-04-23 US disclosed
EP-0529680-B1 Intermediates, their production and their use for preparing alpha-unsaturated amines TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-05-13 EP disclosed
US-5710278-A Herbicidal 1-pyridyltetrazolinones NIHON BAYER AGROCHEM K.K. (JP) 1998-01-20 US disclosed
US-5641727-A Herbicidal 1-pyridyltetrazolinones NIHON BAYER AGROCHEM K.K. (JP) 1997-06-24 US disclosed
EP-0692482-A2 1-pyridyltetrazolinone derivatives NIHON BAYER AGROCHEM K.K. (JP) 1996-01-17 EP disclosed
US-5214152-A Insecticides, miticides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-05-25 US disclosed
US-5175301-A Insecticide, miticide, pesticide TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-29 US disclosed
US-4980357-A ANTIDIABETIC AGENTS PFIZER INC. (US) 1990-12-25 US disclosed
WO-1989001775-A1 AZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1989-03-09 WO disclosed
EP-0306251-A2 Azolidinedione derivatives PFIZER INC. (US) 1989-03-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090280106-A1 Pituitary adenylate cyclase acivating peptide (pacap) receptor (vpac2) agonists and their pharmacological methods of use ADCYAP1R1, VIPR2, ADCY2 P2RX7 620/4885KDM4E 2974/4885TDP1 4059/4885
US-20120015941-A1 Antibacterial Amide and Sulfonamide Substituted Heterocyclic Urea Compounds NAAA, AADAC, RPSA P2RX7 2058/4885KDM4E 1862/4885TDP1 4434/4885
US-20230108636-A1 COMPOSITIONS AND METHODS FOR ENHANCING TRANSPORT THROUGH MUCUS SLC26A4, SLC26A3, SLC10A2 P2RX7 387/4885KDM4E 4800/4885TDP1 4403/4885
US-20090105122-A1 Selective neuropeptide y2 receptor agonists NPY2R, NPY1R, NPY4R P2RX7 297/4885KDM4E 2397/4885TDP1 3566/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.