SCHEMBL3633710

SCHEMBL3633710

CCN(CC)c1ccc(C#CCO)cc1C(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MELK Q14680 1/20 0.39
SLC6A4 P31645 1/20 0.32
MMP2 P08253 1/20 0.31
MMP12 P39900 1/20 0.31
ITK Q08881 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ACACB O00763 1/20 0.30
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA5 P31644 1/20 0.30
GABRA3 P34903 1/20 0.30
GABRA2 P47869 1/20 0.30
GABRB2 P47870 1/20 0.30
GABRA4 P48169 1/20 0.30
GABRE P78334 1/20 0.30
GABRA6 Q16445 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3634001 0.83 CYP1A1 (0.33)
SCHEMBL3722540 0.77 RARA (0.38) MELKSLC6A4MMP2MMP12ALDH1A1
SCHEMBL2099746 0.73 ALDH1A1 (0.41) ALDH1A1GABRA1GABRB1HSP90AA1HSP90AB1
SCHEMBL9532118 0.71 ALDH1A1 (0.45) MMP2MMP12ALDH1A1GABRPGABRD
SCHEMBL12889911 0.71 CRHR1 (0.43) HSP90AA1HSP90AB1KDM4ELMNA
SCHEMBL2098474 0.71 HCAR3 (0.34) HSP90AA1HSP90AB1
SCHEMBL3633553 0.70 MELK (0.34) MELKALDH1A1
SCHEMBL2099560 0.67 HCAR3 (0.43) ACACBHSP90AA1HSP90AB1
SCHEMBL8112207 0.67 ACACB (0.45) MELKMMP2MMP12ACACBGABRP
SCHEMBL2099952 0.66 ALDH1A3 (0.61) ALDH1A1HSP90AA1HSP90AB1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2146951-A2 NOVEL RAR RECEPTOR AGONIST LIGANDS AND USE THEREOF IN HUMAN MEDICINE AND COSMETICS Galderma Research & Development (FR) 2010-01-27 EP disclosed
WO-2008152260-A2 NOVEL RAR RECEPTOR AGONIST LIGANDS AND USE THEREOF IN HUMAN MEDICINE AND COSMETICS GALDERMA RESEARCH & DEVELOPMENT (FR) 2008-12-18 WO disclosed