SCHEMBL363527

SCHEMBL363527

Cc1cc(C2=NOC(c3cc(Cl)cc(Cl)c3)(C(F)(F)F)C2)ccc1C(=O)Cl

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
RXRB P28702 2/20 0.34
RXRA P19793 1/20 0.34
KDM4E B2RXH2 2/20 0.32
RECQL P46063 1/20 0.31
HPGD P15428 1/20 0.31
ORAI1 Q96D31 2/20 0.31
MAPT P10636 1/20 0.31
PKM P14618 1/20 0.30
IL2 P60568 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20261758 1.00 CA1 (0.35) CA1CA2RXRBRXRAKDM4E
SCHEMBL31191610 0.94 RXRA (0.38) CA1CA2RXRBRXRAKDM4E
SCHEMBL29397265 0.92 RXRB (0.41) CA1CA2RXRBRXRAKDM4E
SCHEMBL12274098 0.92 RXRB (0.41) CA1CA2RXRBRXRAKDM4E
SCHEMBL1694737 0.92 CA1 (0.35) CA1CA2RXRBRXRAKDM4E
SCHEMBL362701 0.92 RXRB (0.41) CA1CA2RXRBRXRAKDM4E
SCHEMBL2014009 0.92 RXRB (0.41) CA1CA2RXRBRXRAKDM4E
SCHEMBL29385555 0.92 RXRB (0.41) CA1CA2RXRBRXRAKDM4E
Hydrochloric Acid SCHEMBL1566413 0.91 RXRB (0.40) CA1CA2RXRBRXRAKDM4E
SCHEMBL16243447 0.91 GPR52 (0.38) CA1CA2RXRBRXRAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250214950-A1 METHOD FOR PREPARING FLURALANER HANGZHOU NORMAL UNIVERSITY (CN) 2025-07-03 US disclosed
CN-118930531-A Isoxazoline derivative and preparation method and application thereof 山东省联合农药工业有限公司 2024-11-12 CN disclosed
CN-117800930-A Preparation method of fluororalrana 杭州师范大学 2024-04-02 CN disclosed
US-20230355590-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL CORPORATION (JP) 2023-11-09 US disclosed
US-10874645-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL CORPORATION (JP) 2020-12-29 US disclosed
US-10710991-B2 Process for the preparation of thietane derivatives SYNGENTA PARTICIPATIONS AG (CH) 2020-07-14 US disclosed
US-20200155511-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL CORPORATION (JP) 2020-05-21 US disclosed
US-10596157-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL CORPORATION (JP) 2020-03-24 US disclosed
US-20190315728-A1 PROCESS FOR THE PREPARATION OF THIETANE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2019-10-17 US disclosed
US-10266524-B2 Process for the preparation of thietane derivatives SYNGENTA PARTICIPATIONS AG (CH) 2019-04-23 US disclosed
WO-2010072602-A1 SUBSTITUTED AMIDINE COMPOUNDS FOR COMBATING ANIMAL PESTS BASF SE (DE) 2010-07-01 WO disclosed
US-20100144797-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PEST CONTROL AGENT NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2010-06-10 US disclosed
US-7700808-B2 1-3-bis(substituted phenyl)-3-hydroxypropan-1-one or 2-propen-1-one compound, and salt thereof NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2010-04-20 US disclosed
US-7662972-B2 Isoxazoline-substituted benzamide compound and pesticide NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2010-02-16 US disclosed
EP-2151437-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PEST CONTROL AGENT Nissan Chemical Industries, Ltd. (JP) 2010-02-10 EP disclosed
US-20090312330-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2009-12-17 US disclosed
US-20090023923-A1 1,3-Bis(Substituted Phenyl)-3-Hydroxypropan-1-One or 2-Propen-1-One Compound, and Salt Thereof NISSAN CHEMICAL INDUSTRIES, LTD (JP) 2009-01-22 US disclosed
EP-1975149-A1 1,3-BIS(SUBSTITUTED PHENYL)-3-HYDROXYPROPAN-1-ONE OR 2-PROPEN-1-ONE COMPOUND, AND SALT THEREOF Nissan Chemical Industries, Ltd. (JP) 2008-10-01 EP disclosed
EP-1932836-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND HARMFUL ORGANISM-CONTROLLING AGENT Nissan Chemical Industries, Ltd. (JP) 2008-06-18 EP disclosed
US-20070066617-A1 Insecticidal and acaricidal activity for many agricultural insect pests, spider mites; endo- or ecto-parasiticide for mammals or birds; veterinary medicine; environmentally friendly NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2007-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230355590-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE HDAC7, ACHE, BRDT CA1 1596/4885CA2 377/4885RXRB 1303/4885
US-10596157-B2 Isoxazoline-substituted benzamide compound and pesticide CHRM3, C3AR1, C9 CA1 702/4885CA2 749/4885RXRB 689/4885
US-20100144797-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PEST CONTROL AGENT H1-2, H1-0, H1-3 CA1 1940/4885CA2 431/4885RXRB 1619/4885
US-20090312330-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE ATM, CHRM1, NAT1 CA1 1945/4885CA2 725/4885RXRB 1458/4885
US-10874645-B2 Isoxazoline-substituted benzamide compound and pesticide C3AR1, C5, C9 CA1 916/4885CA2 992/4885RXRB 926/4885
US-20090023923-A1 1,3-Bis(Substituted Phenyl)-3-Hydroxypropan-1-One or 2-Propen-1-One Compound, and Salt Thereof HCN1, CNPY2, CLIC1 CA1 1349/4885CA2 294/4885RXRB 1420/4885
US-10710991-B2 Process for the preparation of thietane derivatives CYP4B1, CYP1B1, CYP1A1 CA1 1180/4885CA2 1260/4885RXRB 2835/4885
US-20190315728-A1 PROCESS FOR THE PREPARATION OF THIETANE DERIVATIVES CYP4B1, CYP1B1, CYP1A1 CA1 1180/4885CA2 1260/4885RXRB 2835/4885
US-20070066617-A1 Insecticidal and acaricidal activity for many agricultural insect pests, spider mites; endo- or ecto-parasiticide for mammals or birds; veterinary medicine; environmentally friendly CHRM1, DDT, ATM CA1 2192/4885CA2 878/4885RXRB 1129/4885
US-20200155511-A1 ISOXAZOLINE-SUBSTITUTED BENZAMIDE COMPOUND AND PESTICIDE C3AR1, C5, C9 CA1 916/4885CA2 992/4885RXRB 926/4885
US-10266524-B2 Process for the preparation of thietane derivatives CYP4B1, CYP1B1, CYP1A1 CA1 1180/4885CA2 1260/4885RXRB 2835/4885
US-20250214950-A1 METHOD FOR PREPARING FLURALANER FFAR4, FFAR2, CYP2A13 CA1 1924/4885CA2 1280/4885RXRB 142/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.