SCHEMBL3650607

SCHEMBL3650607

O=C(O)c1cc(-c2nnn[nH]2)cc(-c2cc(Cl)ccc2Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
ALPL P05186 3/20 0.39
MARS1 P56192 1/20 0.38
SRD5A2 P31213 1/20 0.37
AURKA O14965 2/20 0.37
TPX2 Q9ULW0 2/20 0.37
MAP2K4 P45985 1/20 0.37
HDAC6 Q9UBN7 1/20 0.36
EIF4E P06730 1/20 0.35
F11 P03951 2/20 0.35
CA12 O43570 1/20 0.35
CNR2 P34972 1/20 0.35
CTRC Q99895 1/20 0.35
MAPK1 P28482 1/20 0.34
NOTUM Q6P988 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3653446 0.90 MARS1 (0.49) ALPLMARS1SRD5A2AURKATPX2
SCHEMBL3655999 0.86 ALPL (0.46) TP53ALPLCTRC
SCHEMBL3658838 0.85 KMO (0.41) ALPLMARS1SRD5A2AURKATPX2
SCHEMBL3652824 0.85 ALDH1A1 (0.44) ALDH1A1
SCHEMBL3652199 0.84 CTRC (0.47) ALPLAURKATPX2MAP2K4CA12
SCHEMBL3652133 0.81 CTSA (0.40) ALDH1A1ALPLHDAC6EIF4ECNR2
SCHEMBL3211407 0.81 TSHR (0.42) ALDH1A1ALPLSRD5A2AURKATPX2
SCHEMBL3660881 0.81 AXL (0.38) ALDH1A1ALPLMARS1SRD5A2MAP2K4
SCHEMBL3658374 0.81 EIF4E (0.38) TP53ALPLMARS1SRD5A2MAP2K4
SCHEMBL2513559 0.79 ALOX15 (0.36) ALDH1A1TP53MAP2K4CA12MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205573-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. Hoffmann-Roche AG (CH) 2010-07-14 EP claimed
WO-2009043780-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-04-09 WO claimed
EP-2205573-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009043780-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-04-09 WO disclosed