SCHEMBL365769

SCHEMBL365769

CCOc1ccc(COc2cc(OC(=O)N(C)C)cn3c2c(C(=O)O)c2ccccc23)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 4/20 0.39
LTB4R2 Q9NPC1 4/20 0.39
ALOX5 P09917 1/20 0.38
CNR2 P34972 1/20 0.38
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TP53 P04637 2/20 0.37
PKM P14618 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KMT2A Q03164 4/20 0.36
MEN1 O00255 2/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
S1PR3 Q99500 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365837 0.92 CNR2 (0.37) LTB4RLTB4R2ALOX5CNR2LMNA
SCHEMBL366851 0.91 ALDH1A1 (0.38) LTB4RLTB4R2CNR2TP53ALDH1A1
SCHEMBL365593 0.91 MRGPRX4 (0.39) LTB4RLTB4R2SMN1; SMN2TP53PKM
SCHEMBL365986 0.86 KMT2A (0.38) LTB4RLTB4R2ALOX5CNR2LMNA
SCHEMBL365169 0.84 ACHE (0.41) LTB4RLTB4R2
SCHEMBL366481 0.83 ACHE (0.39) LTB4RLTB4R2SMN1; SMN2TP53MRGPRX4
SCHEMBL366374 0.83 ALDH1A1 (0.38) CNR2LMNAALDH1A1MAPTKMT2A
SCHEMBL365189 0.83 ACHE (0.37) LTB4RLTB4R2CNR2SMN1; SMN2ALDH1A1
SCHEMBL366751 0.83 PPARG (0.33) CNR2ALDH1A1MAPTITGB1ITGA4
SCHEMBL367734 0.82 ATM (0.40) LMNAPKMALDH1A1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed